序号 | 专利名 | 申请号 | 申请日 | 公开(公告)号 | 公开(公告)日 | 发明人 |
---|---|---|---|---|---|---|
61 | JPS6212217B2 - | JP12650278 | 1978-10-14 | JPS6212217B2 | 1987-03-17 | SUGITANI HATSUO; MUKOYAMA YOSHUKI; SONOGASHIRA MIKIO; SONEHARA TAKASHI; MIWA YOJI |
62 | Difluoroketone peptide derivative, manufacture and leucocyte elastase inhibitor | JP13045786 | 1986-06-06 | JPS6253951A | 1987-03-09 | TRAINOR DIANE AMY; STEIN MARK MORRIS |
The invention discloses a series of difluoroketone, mono- di- and tri-peptide derivatives of formula Ia, Ib and Ic: -(Formula set out on pages following Examples) Ia -(Formula set out on pages following Examples) Ib -(Formula set out on pages following Examples) Ic - and salts thereof where appropriate, and wherein the radicals are defined hereafter in the specification. The derivatives are useful in inhibiting the action of human leukocyte elastase. There are also disclosed methods and intermediates for the manufacture of, and pharmaceutical compositions comprising, the said derivatives. | ||||||
63 | Alkene, alkine and cycloalkylene derivative, manufacture andmedicinal composition for treating androgen dependent syndrome | JP3206986 | 1986-02-18 | JPS61189243A | 1986-08-22 | HUGHES LESLIE RICHARD; TUCKER HOWARD |
64 | Substituted phenoxyurea, its preparation, herbicide containing same as an active intredient | JP24804084 | 1984-11-26 | JPS61126065A | 1986-06-13 | HASHIMOTO ISAO; ISHIDA TATSUKAZU; TAKAHASHI KATSUYA; KATO SUSUMU; MIYAZAWA TAKESHIGE; NAKAMURA YASUO |
NEW MATERIAL:A compound of formula I (A is Cl, trifluoromethyl; X, Y, Z are H, Cl, trifluoromethyl; R 1 is 1W6C alkyl, lower alkenyl, lower alkinyl; R 2 is H, 1W6C alkyl). EXAMPLE: 3-(2,5-Dichlorophenoxy)-1,1-dimethylurea. USE: Herbicide: it shows powerful herbicidal effect against annual barnyard grass or prennial bulrush, because it has sufficiently high selectivity to cause no chemical injury to rice plants even when high dose of the chemical is applied. PREPARATION: The reaction of a phenoxyamine of formula II and a carbamoyl halide of formula III (R 2' is 1W6C alkyl, lower alkenyl, etc.) is effected in the presence of a base to give the objective compound of formula IV. COPYRIGHT: (C)1986,JPO&Japio | ||||||
65 | JPS598272B2 - | JP15161775 | 1975-12-17 | JPS598272B2 | 1984-02-23 | YAMAMOTO MICHIHIRO; KOSHIBA MASAO; YAMAMOTO HISAO |
66 | Carbacycline compound and intermediates | JP2226383 | 1983-02-15 | JPS58154521A | 1983-09-14 | POORU ADORIAN ARISUTOFU |
67 | Novel urea derivative and its preparation | JP10927678 | 1978-09-05 | JPS5535067A | 1980-03-11 | TSUJIHARA KENJI; OOZEKI MASAKATSU; ARAI YOSHIHISA |
NEW MATERIAL:A urea derivative of formula I: (R 1 is 1W20C alkyl, 1W6C hydroxyalkyl, 2W5C alkenyl, or 3W5C alkynyl group; R 2 is aldopentofuranosyl; aldopentopyranosyl group, etc.). EXAMPLE: 1-(2-chloroethyl)-3-methyl-3-D-glucopyranosyl urea. USE: An intermediate for the synthesis of 1-(2-chloroethyl)-1-nitroso-3,3-disubstituted urea, having an antitumor action. PROCESS: A secondary amine of formula II is condensed with 2-chloroethyl isocyanate of formula III to give the compound of formula I, which is nitrosated to form the title antitumor compound. COPYRIGHT: (C)1980,JPO&Japio | ||||||
68 | JPS5423720B2 - | JP1998177 | 1977-02-25 | JPS5423720B2 | 1979-08-15 | |
69 | JPS546278B2 - | JP7394777 | 1977-06-23 | JPS546278B2 | 1979-03-27 | |
70 | JPS5328905B2 - | JP12498674 | 1974-10-31 | JPS5328905B2 | 1978-08-17 | |
71 | Polyetherrpolyureido and process for producing same | JP7394777 | 1977-06-23 | JPS532597A | 1978-01-11 | HEINZU SHIYURUTSU |
72 | JPS5249460B2 - | JP12237472 | 1972-12-06 | JPS5249460B2 | 1977-12-17 | |
73 | Preparation of urea derivatives | JP15161775 | 1975-12-17 | JPS5273801A | 1977-06-21 | YAMAMOTO MICHIHIRO; KOSHIBA MASAO; YAMAMOTO HISAO |
PURPOSE: Urea derivatives are easily prepared in good yield by the reaction of N-substd. trihaloacetamide derivatives with ammonia or amines. COPYRIGHT: (C)1977,JPO&Japio | ||||||
74 | JPS506455B1 - | JP2426969 | 1969-03-28 | JPS506455B1 | 1975-03-14 | |
75 | JPS4942830A - | JP8850472 | 1972-09-04 | JPS4942830A | 1974-04-22 | |
76 | JPS4864026A - | JP12237472 | 1972-12-06 | JPS4864026A | 1973-09-05 | |
77 | (메트)아크릴레이트 화합물, 이로부터 유도된 반복단위를 포함하는 코폴리머 및 호모폴리머 | KR1020150136624 | 2015-09-25 | KR101749414B1 | 2017-06-21 | 박광승; 이미린; 박준욱; 허은수; 전성현 |
본명세서는 (메트)아크릴레이트화합물, 이로부터유도된반복단위를포함하는코폴리머및 호모폴리머에관한것이다. | ||||||
78 | 이온성 액체계 촉매 및 이를 이용한 N,N''-치환 우레아의 제조 방법 | KR1020140175291 | 2014-12-08 | KR101644141B1 | 2016-07-29 | 김용진; 트엉꽁지엔; 소정은; 신승한; 조진구 |
본발명은 1 내지 3개의질소원자를갖는 N-헤테로고리구조를포함하는유기계음이온및 그의양이온을포함하는이온성액체계촉매및 이촉매존재하에서아민화합물및 이산화탄소를반응시켜 N,N'-치환우레아를선택적으로제조하는방법에관한것이다. 본발명에서제조되는치환우레아들은모두카바메이트를거쳐이소시아네이트로쉽게전환이가능하고, 이소시아네이트는폴리올과의반응을통해폴리우레탄으로전환될수 있는중요한전구체화합물로사용될수 있다. 한편, 본발명에서의이온성액체계촉매는여러번의재사용이가능하므로경제적이다. | ||||||
79 | 우레아 경화제를 함유하는 저온 경화성 에폭시 조성물 | KR1020100088834 | 2010-09-10 | KR101308611B1 | 2013-09-23 | 아브도우라자크,아테예하우스세인; 베다지,가미니아난다 |
본 발명은 에폭시 수지, 에폭시 경화제, 및 에폭시 경화제에 대한 촉진제의 접촉 생성물을 포함하는 열 경화성 에폭시 조성물로서, 경화제 또는 촉진제가 이소시아네이트와, 하나 이상의 1차 또는 2차 아민 및 두개 이상의 3차 아민을 갖는 하기 화학식의 알킬화된 폴리알킬렌폴리아민의 반응 생성물인 우레아 화합물인 열 경화성 에폭시 조성물에 관한 것이다:
상기 식에서, R 1 , R 2 , R 3 , R 4 및 R 5 는 독립적으로 수소, 메틸 또는 에틸이고, n 및 m은 독립적으로 1 내지 6의 정수이고, X는 1 내지 10의 정수이다. |
||||||
80 | 지방족 디우레아의 제조방법 | KR1020100008396 | 2010-01-29 | KR1020110088749A | 2011-08-04 | 김훈식; 정민석; 누엔딘콴; 심유나 |
PURPOSE: A method for manufacturing aliphatic diurea is provided to prepare diurea with high yield and high selectivity in a mild condition using water as a reaction solvent and catalyst and to simplify a refining process of products. CONSTITUTION: A method for manufacturing aliphatic diurea comprises a step of reacting C2-8 aliphatic diamine with urea to prepare aliphatic diurea using water as a reaction solvent and a catalyst. The C2-8 aliphatic diamine is 1,2-ethanediamine, 1,3-propanediamine, 1,4-butanediamine, 1,6-hexanediamine, 1,8-octane diamine, 1,2-cyclohexane diamine, 1,3-cyclohexanediamine, 1,4-cyclohexanediamine, 1,3-cyclohexane bismethylamine or 1,4-cyclohexane bismethylamine. |