161 |
Acid-cleavable compound, positive type radiation-sensitive mixture containing the same, and radiation-sensitive recording material produced with the said mixture |
JP12407792 |
1992-04-17 |
JPH05194357A |
1993-08-03 |
GEORUKU PAUROSUKII; HORUSUTO RESHIERUTO; WARUTAA SHIYUPIISU; RARUFU DAMERU |
PURPOSE: To provide the new compounds useful as radiation-sensitive recording materials showing a high resolution and high image contrast.
CONSTITUTION: The compounds of the formula (R
1 is an alkylene, cycloalkylene, alkenylene, etc.; R
2 is an alkyl, alkenyl, cycloalkyl, aryl, etc.; R
3 is an alkyl, aryl; X is -CO-, -O-CO-, -NH-CO-; (n) ≥2, particularly 3 to 50) are obtained, for example, by reacting benzaldehyde dimethylacetal with urethane-alcohol in toluene in the presence of p-toluenesufonic acid. The compounds are cleavable by acid and, in combination with photolytic acid donors and alkali-soluble binders, are constituents of positive type mixtures, which are used particularly for recording materials for UV radiation and high energy radiation.
COPYRIGHT: (C)1993,JPO |
162 |
Glycolic acid derivative |
JP15415491 |
1991-03-15 |
JPH0532609A |
1993-02-09 |
PEETAA RADATSUTSU; KURAUSU YOTSUTO SHIYUMITSUCHIE; KURAUSUUOTSUTOO MINKU |
PURPOSE: To provide a new glycolic acid derivative and its salt usable as medicinally active substance for disease of cardia, circulatory organ and blood vessel, especially for prevention and treatment of hypertension, cardiac incompetence and high aldosteronism.
CONSTITUTION: The derivs. of glycolic acid represented by formula [where X is R
8, R
8-O-C
mH
2m-CO- ((m) is 0-10), R
8-SO
2-R
9R
10N-C
mH
2m-CO-, etc.; R
1, R
3, R
6, R
7, R
9 and R
10 are H, A (A is a 1-8 alkyl); R
2, R
4 and R
8 are H, A, Ar, Ar-alkyl, Het (Het is a 5- or 6-membered heterocyclicring); R
5 is (H, OH), (H, NH
2) or =O; Y is 0 or 1 of residual group of amino acid selected from among Abu, Ada, Ala, Bia, etc.; Z is -CN, etc.] and the salts thereof, e.g. N-[2- isopropyl-4-hydroxy-5-(4-aminopiperidinocarbonyl-Pla-His-amino)-6- cyclohexylhexyl]-propanesulfonamide. The compd. represented by formula I is obtained, for example by treating a kind of derivative of the compd. represented by formula I having a functional group with a solvolysis agent, etc.
COPYRIGHT: (C)1993,JPO |
163 |
JPH04500377A - |
JP50614189 |
1989-05-30 |
JPH04500377A |
1992-01-23 |
|
|
164 |
JPH0322873B2 - |
JP19055487 |
1987-07-31 |
JPH0322873B2 |
1991-03-27 |
ROOZUMARII TEPUFURU; IERUKU BINSU |
|
165 |
JPH0147461B2 - |
JP13700580 |
1980-09-29 |
JPH0147461B2 |
1989-10-13 |
NODA KANJI; NAKAGAWA AKIRA; MOTOMURA TOSHIHARU; MYATA SATORU; INOE TOSHITAKA; IDE HIROYUKI |
|
166 |
Enantiomer of bicyclo(4,2,0)oct-2-ene-7-one, novel synthesis of derivatives of same and bicyclo(4,2,0)octane derivatives and intermediate therefor |
JP21000687 |
1987-08-24 |
JPS6393742A |
1988-04-25 |
AASAA EFU KURATSUGU; DENISU JIEI KAATESUZU |
|
167 |
Multifunctional carbodiimide having specific structure |
JP23471286 |
1986-10-03 |
JPS6391356A |
1988-04-22 |
JIEIMUZU UEIN TEIRAA |
|
168 |
Peptide compound |
JP20862186 |
1986-09-04 |
JPS6363649A |
1988-03-22 |
MORISAWA YASUHIRO; YABE YUICHIRO; KATAOKA MITSURU; IIJIMA YASUTERU; TAKAHAGI HIDEKUNI; KOKUBU TATSURO; HIWADA KUNIO |
NEW MATERIAL:The compound of formula I [R<1> is -B-R<7> (B is lower alkylene; R<7> is aryl, etc.), etc., R<2> is aryl or heteroaryl; R is H or lower alkyl; R<3> is H, 1-10C alkyl, etc.; R<4> is isopropyl, phenyl, etc.; R<5> is 1-5C alkyl; R<6> is substituted 1-10C alkyl, etc.]. EXAMPLE:N<alpha>-[bis(1-naphthylmethyl)acetyl]-L-histidyl-statyl-L-leu cyl-epsilon-L-lysinol. USE:A renin inhibitor useful as a diagnostic and remedy for hypertension. PREPARATION:The compound of formula I can be produced by reacting the compound of formula II (R<3>a is R<3> having protected amino, carboxy, etc., or same as R<3>) with the compound of formula III (R<6>a is R<6> having protected amino, guanidyl, etc., or same as R<6>) and deprotecting the resultant product. |
169 |
JPS637088B2 - |
JP15018382 |
1982-08-31 |
JPS637088B2 |
1988-02-15 |
JON UINFURITSUDO AGAA |
|
170 |
JPS636544B2 - |
JP564479 |
1979-01-23 |
JPS636544B2 |
1988-02-10 |
HANSU YOAHIMU HENIHI; PEETERU TSUIIMEKU; ERUHARUTO SHERUMAN |
|
171 |
Manufacture of trans-cyclohexane-1,4-diisocyanate |
JP1743587 |
1987-01-29 |
JPS62246547A |
1987-10-27 |
HANSU TSUENGERU; MANFUREETO BERUKUFUERUTO |
|
172 |
JPS6241496B2 - |
JP1597079 |
1979-02-16 |
JPS6241496B2 |
1987-09-03 |
KOMATSU KAZUO; MATSUMOTO SOJIRO; MANIWA TAKESHI; NIIMURA NOBUYUKI |
|
173 |
Ethanol amine derivative |
JP24514886 |
1986-10-15 |
JPS62174041A |
1987-07-30 |
HARII FUINCHI; ROORENSU HENRII CHIYAARUZU RAN; ARAN NAIRAA; IAN FUREDERITSUKU SUKITSUDOMOA; IAN BAKUSUTAA KIYANBERU; DEIBITSUDO MIDORUMISU; CHIYAARUZU UIRUBII |
|
174 |
Ureidorennin inhibitor |
JP31611886 |
1986-12-23 |
JPS62164658A |
1987-07-21 |
SESHIYA IERU NATARAJIYAN; DENISU EBAN RIONO; EDOWAADO UIRIAMU PETORIIRO JIY |
Compounds of the formula are disclosed wherein: X may comprise an amino acid such as Phe, His or Trp; R4, R1 and R9 are side chains of amino acids such as His, Ile, Phe and Val; and q may be zero or one. These compounds intervene in the conversion of angiotensinogen to angiotensin II by inhibiting renin and thus are useful as anti-hypertensive agents. |
175 |
JPS6229425B2 - |
JP2759778 |
1978-03-10 |
JPS6229425B2 |
1987-06-25 |
HANSU TSUENGERU; MANFUREETO BERUKUFUERUTO |
|
176 |
(meth)acrylic acid esters |
JP14314786 |
1986-06-20 |
JPS61293960A |
1986-12-24 |
IENSU BINKERU; BURUUNO BEEMAA; KARURU HANSU ZUYURINGU; YURUGEN RAINAASU; BORUFUGANGU POTSUTSUN |
|
177 |
JPS6136508B2 - |
JP7877978 |
1978-06-30 |
JPS6136508B2 |
1986-08-19 |
KURAUSU KEENIHI; UORUFUGANGU RAIHIMAN; YOOZEFU PEDAIN |
|
178 |
Fluorochemical allophanate |
JP13885585 |
1985-06-25 |
JPS6124557A |
1986-02-03 |
RICHIYAADO MAAKU SUTAAN |
|
179 |
JPS6053017B2 - |
JP1864778 |
1978-02-22 |
JPS6053017B2 |
1985-11-22 |
HANSU DEIITAA UINKERUMAN; KAARU HAINTSU UORUFU; HARARUDO EERUTERU; NORUBERUTO WAIMAN |
|
180 |
Manufacture of carbamic acid derivative |
JP2660985 |
1985-02-15 |
JPS60199868A |
1985-10-09 |
JIERAARU BARUSERO; JIYAN PIEERU SENE; JIERAARU SANNIE |
|