序号 专利名 申请号 申请日 公开(公告)号 公开(公告)日 发明人
161 Acid-cleavable compound, positive type radiation-sensitive mixture containing the same, and radiation-sensitive recording material produced with the said mixture JP12407792 1992-04-17 JPH05194357A 1993-08-03 GEORUKU PAUROSUKII; HORUSUTO RESHIERUTO; WARUTAA SHIYUPIISU; RARUFU DAMERU
PURPOSE: To provide the new compounds useful as radiation-sensitive recording materials showing a high resolution and high image contrast. CONSTITUTION: The compounds of the formula (R 1 is an alkylene, cycloalkylene, alkenylene, etc.; R 2 is an alkyl, alkenyl, cycloalkyl, aryl, etc.; R 3 is an alkyl, aryl; X is -CO-, -O-CO-, -NH-CO-; (n) ≥2, particularly 3 to 50) are obtained, for example, by reacting benzaldehyde dimethylacetal with urethane-alcohol in toluene in the presence of p-toluenesufonic acid. The compounds are cleavable by acid and, in combination with photolytic acid donors and alkali-soluble binders, are constituents of positive type mixtures, which are used particularly for recording materials for UV radiation and high energy radiation. COPYRIGHT: (C)1993,JPO
162 Glycolic acid derivative JP15415491 1991-03-15 JPH0532609A 1993-02-09 PEETAA RADATSUTSU; KURAUSU YOTSUTO SHIYUMITSUCHIE; KURAUSUUOTSUTOO MINKU
PURPOSE: To provide a new glycolic acid derivative and its salt usable as medicinally active substance for disease of cardia, circulatory organ and blood vessel, especially for prevention and treatment of hypertension, cardiac incompetence and high aldosteronism. CONSTITUTION: The derivs. of glycolic acid represented by formula [where X is R 8, R 8-O-C mH 2m-CO- ((m) is 0-10), R 8-SO 2-R 9R 10N-C mH 2m-CO-, etc.; R 1, R 3, R 6, R 7, R 9 and R 10 are H, A (A is a 1-8 alkyl); R 2, R 4 and R 8 are H, A, Ar, Ar-alkyl, Het (Het is a 5- or 6-membered heterocyclicring); R 5 is (H, OH), (H, NH 2) or =O; Y is 0 or 1 of residual group of amino acid selected from among Abu, Ada, Ala, Bia, etc.; Z is -CN, etc.] and the salts thereof, e.g. N-[2- isopropyl-4-hydroxy-5-(4-aminopiperidinocarbonyl-Pla-His-amino)-6- cyclohexylhexyl]-propanesulfonamide. The compd. represented by formula I is obtained, for example by treating a kind of derivative of the compd. represented by formula I having a functional group with a solvolysis agent, etc. COPYRIGHT: (C)1993,JPO
163 JPH04500377A - JP50614189 1989-05-30 JPH04500377A 1992-01-23
164 JPH0322873B2 - JP19055487 1987-07-31 JPH0322873B2 1991-03-27 ROOZUMARII TEPUFURU; IERUKU BINSU
165 JPH0147461B2 - JP13700580 1980-09-29 JPH0147461B2 1989-10-13 NODA KANJI; NAKAGAWA AKIRA; MOTOMURA TOSHIHARU; MYATA SATORU; INOE TOSHITAKA; IDE HIROYUKI
166 Enantiomer of bicyclo(4,2,0)oct-2-ene-7-one, novel synthesis of derivatives of same and bicyclo(4,2,0)octane derivatives and intermediate therefor JP21000687 1987-08-24 JPS6393742A 1988-04-25 AASAA EFU KURATSUGU; DENISU JIEI KAATESUZU
167 Multifunctional carbodiimide having specific structure JP23471286 1986-10-03 JPS6391356A 1988-04-22 JIEIMUZU UEIN TEIRAA
168 Peptide compound JP20862186 1986-09-04 JPS6363649A 1988-03-22 MORISAWA YASUHIRO; YABE YUICHIRO; KATAOKA MITSURU; IIJIMA YASUTERU; TAKAHAGI HIDEKUNI; KOKUBU TATSURO; HIWADA KUNIO
NEW MATERIAL:The compound of formula I [R<1> is -B-R<7> (B is lower alkylene; R<7> is aryl, etc.), etc., R<2> is aryl or heteroaryl; R is H or lower alkyl; R<3> is H, 1-10C alkyl, etc.; R<4> is isopropyl, phenyl, etc.; R<5> is 1-5C alkyl; R<6> is substituted 1-10C alkyl, etc.]. EXAMPLE:N<alpha>-[bis(1-naphthylmethyl)acetyl]-L-histidyl-statyl-L-leu cyl-epsilon-L-lysinol. USE:A renin inhibitor useful as a diagnostic and remedy for hypertension. PREPARATION:The compound of formula I can be produced by reacting the compound of formula II (R<3>a is R<3> having protected amino, carboxy, etc., or same as R<3>) with the compound of formula III (R<6>a is R<6> having protected amino, guanidyl, etc., or same as R<6>) and deprotecting the resultant product.
169 JPS637088B2 - JP15018382 1982-08-31 JPS637088B2 1988-02-15 JON UINFURITSUDO AGAA
170 JPS636544B2 - JP564479 1979-01-23 JPS636544B2 1988-02-10 HANSU YOAHIMU HENIHI; PEETERU TSUIIMEKU; ERUHARUTO SHERUMAN
171 Manufacture of trans-cyclohexane-1,4-diisocyanate JP1743587 1987-01-29 JPS62246547A 1987-10-27 HANSU TSUENGERU; MANFUREETO BERUKUFUERUTO
172 JPS6241496B2 - JP1597079 1979-02-16 JPS6241496B2 1987-09-03 KOMATSU KAZUO; MATSUMOTO SOJIRO; MANIWA TAKESHI; NIIMURA NOBUYUKI
173 Ethanol amine derivative JP24514886 1986-10-15 JPS62174041A 1987-07-30 HARII FUINCHI; ROORENSU HENRII CHIYAARUZU RAN; ARAN NAIRAA; IAN FUREDERITSUKU SUKITSUDOMOA; IAN BAKUSUTAA KIYANBERU; DEIBITSUDO MIDORUMISU; CHIYAARUZU UIRUBII
174 Ureidorennin inhibitor JP31611886 1986-12-23 JPS62164658A 1987-07-21 SESHIYA IERU NATARAJIYAN; DENISU EBAN RIONO; EDOWAADO UIRIAMU PETORIIRO JIY
Compounds of the formula are disclosed wherein: X may comprise an amino acid such as Phe, His or Trp; R4, R1 and R9 are side chains of amino acids such as His, Ile, Phe and Val; and q may be zero or one. These compounds intervene in the conversion of angiotensinogen to angiotensin II by inhibiting renin and thus are useful as anti-hypertensive agents.
175 JPS6229425B2 - JP2759778 1978-03-10 JPS6229425B2 1987-06-25 HANSU TSUENGERU; MANFUREETO BERUKUFUERUTO
176 (meth)acrylic acid esters JP14314786 1986-06-20 JPS61293960A 1986-12-24 IENSU BINKERU; BURUUNO BEEMAA; KARURU HANSU ZUYURINGU; YURUGEN RAINAASU; BORUFUGANGU POTSUTSUN
177 JPS6136508B2 - JP7877978 1978-06-30 JPS6136508B2 1986-08-19 KURAUSU KEENIHI; UORUFUGANGU RAIHIMAN; YOOZEFU PEDAIN
178 Fluorochemical allophanate JP13885585 1985-06-25 JPS6124557A 1986-02-03 RICHIYAADO MAAKU SUTAAN
179 JPS6053017B2 - JP1864778 1978-02-22 JPS6053017B2 1985-11-22 HANSU DEIITAA UINKERUMAN; KAARU HAINTSU UORUFU; HARARUDO EERUTERU; NORUBERUTO WAIMAN
180 Manufacture of carbamic acid derivative JP2660985 1985-02-15 JPS60199868A 1985-10-09 JIERAARU BARUSERO; JIYAN PIEERU SENE; JIERAARU SANNIE
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