| 序号 | 专利名 | 申请号 | 申请日 | 公开（公告）号 | 公开（公告）日 | 发明人 |
|---|---|---|---|---|---|---|
| 1 | 环丙烷化的大环酮和内酯 | CN200610079337.1 | 2006-04-14 | CN1865257A | 2006-11-22 | A·P·S·纳鲁拉; E·M·阿鲁达; F·T·希特 |
| 本发明涉及一种具有以下通式的新的环丙烷化大环酮和内酯化合物，其中X是选自O、N、S、CH或CH2的原子或官能团；其中Y是由1到20个碳原子组成的直链或支链烃基部分；其中W是由1到20个碳原子组成的直链或支链烃基部分；其中O是氧原子；及这些新化合物在制造香料和香味产品如香水、古龙水和个人护理产品上的用途。 | ||||||
| 2 | Cyclopropanated macrocyclic ketones and lactones | US12329112 | 2008-12-05 | US07943560B2 | 2011-05-17 | Anubhav P.S. Narula; Edward Mark Arruda; Franc T. Schiet |
| The present invention is directed to novel cyclopropanated macrocyclic ketone and lactone compounds of the general formula: wherein X is an atom or a functional group selected from the group consisting of O, N, S, R—CH, and CH2; wherein R is a C1-C3 alkyl group; wherein Y and W independently represent is a linear or branched alkyl or alkenyl group, optionally substituted, consisting of less than 10 and preferably less than 7 carbon atoms; and wherein O is an oxygen atom, and the use of these novel compounds in creating fragrances and scents in items such as perfumes, colognes, and personal care products. | ||||||
| 3 | Cyclopropanated macrocyclic ketones and lactones | US11386957 | 2006-03-22 | US20060234885A1 | 2006-10-19 | Anubhav Narula; Edward Arruda; Franc Schiet |
| The present invention is directed to novel cyclopropanated macrocyclic ketone and lactone compounds of the general formula wherein X is an atom or a functional group selected from the group consisting of O, N, S, CH, or CH2; wherein Y is a straight or branched hydrocarbon moiety consisting of 1 to 20 carbon atoms; wherein W is a straight or branched hydrocarbon moiety of consisting of 1 to 20 carbon atoms; and wherein O is an oxygen atom; and the use of these novel compounds in creating fragrances, and scents in items such as perfumes, colognes and personal care products. | ||||||
| 4 | α-GLUCOSIDASE INHIBITOR | JP2006324346 | 2006-11-30 | JP2008137925A | 2008-06-19 | OZAKI MAKOTO; OE HIROMI; KITAMURA SHINICHI |
| <P>PROBLEM TO BE SOLVED: To provide a new α-glucosidase inhibitor having high activity. <P>SOLUTION: The compound represented by the general formula is extracted from the root and/or above-ground part of Salacia reticulata. <P>COPYRIGHT: (C)2008,JPO&INPIT | ||||||
| 5 | α- glucosidase inhibitor | JP2006324346 | 2006-11-30 | JP4125768B2 | 2008-07-30 | 進一 北村; 弘美 大江; 誠 小崎 |
| 6 | Suppressing methods and compositions of the 5α- reductase activity | JP50328694 | 1993-04-30 | JPH08501771A | 1996-02-27 | リャオ，シューツン; リャン，テーミン |
| (57)【要約】 本明細書において、飽和および不飽和脂肪酸類、その誘導体と合成類縁物質を含む新規クラスの抗アンドロゲン化合物類、その合成方法、およびアンドロゲン活性に起因する疾患の治療へのこれらの化合物の使用を開示する。 さらにまた、抗アンドロゲン活性があることがこれまで分からなかった公知の化合物の、アンドロゲン活性に起因する疾患の治療における使用も開示する。 | ||||||
| 7 | METHODS AND COMPOSITIONS FOR INHIBITING 5$g(a)-REDUCTASE ACTIVITY | EP93910950.0 | 1993-04-30 | EP0652749A1 | 1995-05-17 | LIAO, Shutsung; LIANG, Tehming |
| Disclosed is a novel class of antiandrogenic compounds including saturated and unsaturated fatty acids, their derivatives, and synthetic analogs, their method of synthesis, and their use in treating disorders associated with androgenic activities. Also disclosed is the use of known compounds not previously known for their antiandrogenic activity in treating disorders related to androgenic activities. | ||||||
| 8 | Cyclopropanated macrocyclic ketones and lactones | US12329091 | 2008-12-05 | US07943559B2 | 2011-05-17 | Anubhav P. S. Narula; Edward Mark Arruda; Franc T. Schiet |
| The present invention is directed to novel cyclopropanated macrocyclic ketone and lactone compounds of the general formula: wherein X is an atom or a functional group selected from the group consisting of O, N, S, R—CH, and CH2; wherein R is a C1-C3 alkyl group; wherein Y and W independently represent is a linear or branched alkyl or alkenyl group, optionally substituted, consisting of less than 10 and preferably less than 7 carbon atoms; and wherein O is an oxygen atom, and the use of these novel compounds in creating fragrances and scents in items such as perfumes, colognes, and personal care products. | ||||||
| 9 | Cyclopropanated Macrocyclic Ketones and Lactones | US11674523 | 2007-02-13 | US20070142253A1 | 2007-06-21 | Anubhav Narula; Edward Arruda; Franc Schiet |
| The present invention is directed to novel cyclopropanated macrocyclic ketone and lactone compounds of the general formula wherein X is an atom or a functional group selected from the group consisting of O, N, S, R—CH, CH2 and wherein R is a C1-C3 alkyl group; a wherein Y and W independently represent is a linear or branched alkyl or alkenyl group, possibly substituted, consisting of less than 10 and preferably less than 7 carbon atoms; and wherein O is an oxygen atom; and the use of these novel compounds in creating fragrances, and scents in items such as perfumes, colognes and personal care products. | ||||||
| 10 | Cyclopropanated macrocyclic ketones and lactones | US11105626 | 2005-04-14 | US07189881B2 | 2007-03-13 | Anubhav P. S. Narula; Edward Mark Arruda; Franc T. Schiet |
| The present invention is directed to novel cyclopropanated macrocyclic ketone and lactone compounds of the general formula wherein X is an atom or a functional group selected from the group consisting of O, N, S, CH, or CH2; wherein Y is a straight or branched hydrocarbon moiety consisting of 1 to 20 carbon atoms; wherein W is a straight or branched hydrocarbon moiety of consisting of 1 to 20 carbon atoms; and wherein O is an oxygen atom; and the use of these novel compounds in creating fragrances, and scents in items such as perfumes, colognes and personal care products. | ||||||
| 11 | Methods and compositions for inhibiting 5.alpha.-reductase activity | US904443 | 1992-07-01 | US5422371A | 1995-06-06 | Shutsung Liao; Tehming Liang |
| Disclosed are a novel class of anti-androgenic compounds including saturated and unsaturated fatty acids, their derivatives, and synthetic analogs, according to the following formula:CH.sub.3 --(CH.sub.2).sub.a --(CR.sub.1 R.sub.2 CH.dbd.CH).sub.b --(CH.sub.2).sub.c --COOH,wherein R.sub.1 and R.sub.2 are each either hydrogen or a halogen; wherein a and c are integers from 0-9; wherein b is an integer from 1-6, provided that12<a+c+(3.times.b).ltoreq.22.Also disclose are methods of synthesis of these compounds, and their use in treating disorders associated with androgenic activities. Also disclosed is the use of known compounds not previously known for their anti-androgenic activity in treating disorders related to androgenic activities. | ||||||
| 12 | Tricyclic cage compounds, their synthesis and use as antiviral agents | US171109 | 1980-07-22 | US4347254A | 1982-08-31 | Junki Katsube; Hiromi Shimomura; Shun Inokuma; Akihiko Sugie |
| A compound of the formula: ##STR1## wherein A.sub.1 is a single bond or a C.sub.1 -C.sub.5 alkylene group bonding at the 2-, 2'- or 3-position, A.sub.2 is a C.sub.1 -C.sub.3 alkylene group, A.sub.3 is a C.sub.1 -C.sub.4 alkylene group, X is --O-- or --SO.sub.n -- and B is a carboxy group, a C.sub.2 -C.sub.5 alkoxycarbonyl group, a cyano group, an amino group of the formula: ##STR2## or a carbamoyl group of the formula: ##STR3## which is useful as an antiviral agent with no side effect. | ||||||
| 13 | Cyclopropanated Macrocyclic Ketones and Lactones | US12329112 | 2008-12-05 | US20090087402A1 | 2009-04-02 | Anubhav P.S. Narula; Edward Mark Arruda; Franc T. Schiet |
| The present invention is directed to novel cyclopropanated macrocyclic ketone and lactone compounds of the general formula: wherein X is an atom or a functional group selected from the group consisting of O, N, S, R—CH, and CH2; wherein R is a C1-C3 alkyl group; wherein Y and W independently represent is a linear or branched alkyl or alkenyl group, optionally substituted, consisting of less than 10 and preferably less than 7 carbon atoms; and wherein O is an oxygen atom, and the use of these novel compounds in creating fragrances and scents in items such as perfumes, colognes, and personal care products. | ||||||
| 14 | CYCLOPROPANATED MACROCYCLIC KETONES AND LACTONES | US12329091 | 2008-12-05 | US20090081150A1 | 2009-03-26 | Anubhav P.S. Narula; Edward Mark Arruda; Franc T. Schiet |
| The present invention is directed to novel cyclopropanated macrocyclic ketone and lactone compounds of the general formula: wherein X is an atom or a functional group selected from the group consisting of O, N, S, R—CH, and CH2; wherein R is a C1-C3 alkyl group; wherein Y and W independently represent is a linear or branched alkyl or alkenyl group, optionally substituted, consisting of less than 10 and preferably less than 7 carbon atoms; and wherein O is an oxygen atom, and the use of these novel compounds in creating fragrances and scents in items such as perfumes, colognes, and personal care products. | ||||||
| 15 | Cyclopropanated macrocyclic ketones and lactones | US11386957 | 2006-03-22 | US07485668B2 | 2009-02-03 | Anubhav P. S. Narula; Edward Mark Arruda; Franc T. Schiet |
| The present invention is directed to novel cyclopropanated macrocyclic ketone and lactone compounds of the general formula wherein X is an atom or a functional group selected from the group consisting of O, N, S, CH, or CH2; wherein Y is a straight or branched hydrocarbon moiety consisting of 1 to 20 carbon atoms; wherein W is a straight or branched hydrocarbon moiety of consisting of 1 to 20 carbon atoms; and wherein O is an oxygen atom; and the use of these novel compounds in creating fragrances, and scents in items such as perfumes, colognes and personal care products. | ||||||
| 16 | Cyclopropanated macrocyclic ketones and lactones | US11674523 | 2007-02-13 | US07482380B2 | 2009-01-27 | Anubhav P. S. Narula; Edward Mark Arruda; Franc T. Schiet |
| The present invention is directed to novel cyclopropanated macrocyclic ketone and lactone compounds of the general formula wherein X is an atom or a functional group selected from the group consisting of O, N, S, R—CH, CH2 and wherein R is a C1-C3 alkyl group; a wherein Y and W independently represent is a linear or branched alkyl or alkenyl group, possibly substituted, consisting of less than 10 and preferably less than 7 carbon atoms; and wherein O is an oxygen atom; and the use of these novel compounds in creating fragrances, and scents in items such as perfumes, colognes and personal care products. | ||||||
| 17 | Cyclopropanated macrocyclic ketones and lactones | US11105626 | 2005-04-14 | US20060234883A1 | 2006-10-19 | Anubhav Narula; Edward Arruda; Franc Schiet |
| The present invention is directed to novel cyclopropanated macrocyclic ketone and lactone compounds of the general formula wherein X is an atom or a functional group selected from the group consisting of 0, N, S, CH, or CH2; wherein Y is a straight or branched hydrocarbon moiety consisting of 1 to 20 carbon atoms; wherein W is a straight or branched hydrocarbon moiety of consisting of 1 to 20 carbon atoms; and wherein O is an oxygen atom; and the use of these novel compounds in creating fragrances, and scents in items such as perfumes, colognes and personal care products. | ||||||
| 18 | Propargylic and allenic sulfones | US470814 | 1990-01-26 | US5237101A | 1993-08-17 | K. C. Nicolaou; Guido Zaccarello; Golfo Skokotas; Peter Maligres |
| Propargylic and allenic sulfones are disclosed having the ability to selectively cleave nucleic acids, especially deoxyribonucleic acid. Such compositions are capable of being synthetically modified to effect cleavage at selected, sequenced sites on nucleic acids. | ||||||
| 19 | METHODS AND COMPOSITIONS FOR INHIBITING 5-g(a)-REDUCTASE ACTIVITY. | EP93910950 | 1993-04-30 | EP0652749A4 | 1997-04-09 | LIAO SHUTSUNG; LIANG TEHMING |
| Disclosed are a novel class of anti-androgenic compounds including saturated and unsaturated fatty acids, their derivatives, and synthetic analogs, according to the following formula: CH3-(CH2)a-(CR1R2CH=CH)b-(CH2)c-COOH, wherein R1 and R2 are each either hydrogen or a halogen; wherein a and c are integers from 0-9; wherein b is an integer from 1-6, provided that 12 | ||||||
| 20 | Heterotricyclic compounds, processes for their production and pharmaceutical compositions containing them | EP79300617.2 | 1979-04-12 | EP0006283B1 | 1983-01-26 | Katsube, Junki; Shimomura, Hiromi; Inokuma, Shun; Sugie, Akihiko |
QQ群二维码
意见反馈
意见反馈