| 序号 | 专利名 | 申请号 | 申请日 | 公开（公告）号 | 公开（公告）日 | 发明人 |
|---|---|---|---|---|---|---|
| 61 | D1 piperidinyl replacement methanolate anthracene as an antagonist / d2 antagonists and 5ht2- serotonin antagonist | JP50389395 | 1994-07-04 | JP3031634B2 | 2000-04-10 | クリマス，マイケル・サデウス; タープコ，マーク・オーナル |
| 62 | JPH05508832A - | JP50800191 | 1991-04-03 | JPH05508832A | 1993-12-09 | |
| 63 | Heribicide | JP25719189 | 1989-10-03 | JPH02149567A | 1990-06-08 | PIITAA SUCHIYUAATO GEITSU; GUREIAMU PIITAA JIYOONZU |
| NEW MATERIAL: Sulfone anilide of formula I (wherein A is N or CR 5; X is O or S; Y is N or CR 9 is alkyl, alkenyl, alkynyl, cycloalkyl, aryl, heterocycle, etc.; R 2 is H, alkyl, carboxylic acid acyl, etc.; R 3 and R 4 are each H, alkyl, alkoxy, cycloalkyl, etc.; R 6, R 7 and R 8 are each H, halogen, cyano, etc.; and R 5 is similar to R 6-R 8 or aryloxy or heterocycle-oxy; and R 9 is H or alkyl) and its salt. EXAMPLE: 2'-Chloro-6'-(4,6-dimethoxy-2-pyrimidinyloxy)-1,1,1-trifluoromethane sulfone anilide. USE: Herbicides, safe for grain, wheat, etc., weeding selectively. PROCESS: For example, an anilide corresponding to aniline of formula II is reacted with a compound of formula III to obtain a compound of formula I. COPYRIGHT: (C)1990,JPO | ||||||
| 64 | Novel derivative of 1-dithia-2-thiacephalosporanic acid, its production, use thereof as drug and pharmaceutical composition containing the same | JP2407788 | 1988-02-05 | JPS63253088A | 1988-10-20 | JIYOZEFU AZODEI; SORANJIYU GOWAN DANBURIEERU; JIYANJIYORUJIYU TOUUCHI |
| 65 | Thieno-1, 4-diazepine | JP1120487 | 1987-01-20 | JPS62181282A | 1987-08-08 | BERUNAA SUTORANSUKII; KAARU HAINTSU UEEBAA; GERUHARUTO BUARUSAA; ARUBUREHITO HAREUSU; YORUGE KASARUZU SUTENTSUERU; GOYUKO MUASEBITSUKU; BUORUFU DEIITORITSUHI BETSUKUT |
| 66 | JPS62500591A - | JP50482585 | 1985-10-22 | JPS62500591A | 1987-03-12 | |
| 67 | JPS6056159B2 - | JP17994880 | 1980-12-18 | JPS6056159B2 | 1985-12-09 | GOTO KYOTO; TSUDA YOSHIAKI; DOI TADAHIRO |
| 68 | JPS60500912A - | JP50154284 | 1984-03-21 | JPS60500912A | 1985-06-20 | |
| 69 | Thiazolobenzoxazine derivatives and process for preparing same | JP1304876 | 1976-02-09 | JPS5295696A | 1977-08-11 | MATSUDA HIDEAKI; KURAISHI TADAYUKI; KATORI TATSUHIKO; OONO HIROMITSU; ODAKA YOSHICHIKA |
| 70 | 비정형적인 향정신성 작용을 갖는피롤로[2,1-ｂ][1,3]벤조티아제핀 | KR1020017001214 | 1999-07-27 | KR100642730B1 | 2006-11-03 | 캄피아니기우스페; 나치비토; 미네티파트리샤; 디세사르마리아아순타 |
| 다음 화학식 1의 피롤로[2,1-b][1,3]벤조티아제핀 구조에 대한 새로운 축합중합된 이종고리는 설명에 나타내 것과 같은 것으로써 정의된다. 알려진 정신병 치료제와 비교하여 본 발명에 따른 화합물의 실질적인 작용은 원치않는 추체외로의 증상을 감소시킴과 관련되어 있다. 본 발명의 화합물은 정신분열증과 같은 정신병의 치료를 위한 약제학적 조성물의 형태를 가질 것이다. 화학식 1 정신병 치료제, 비정형적인, 피롤로[2,1-b][1,3]벤조티아제핀 | ||||||
| 71 | 두고리 피리미딘-5-온 유도체의 제조방법 | KR1019820002847 | 1982-06-25 | KR100023836B1 | 1987-07-20 | 루우도이.제이케니이스; 죠셉스씨.마아텐스 |
| 72 | 두고리 피리미딘-5-온 유도체의 제조방법 | KR1019820002847 | 1982-06-25 | KR1019840000568A | 1984-02-25 | 루우도이.제이케니이스; 죠셉스씨.마아텐스 |
| 내용없음 | ||||||
| 73 | 3,5-디-3급- 부틸 -4- 하이드록시 페닐-치환 복소환 화합물의 제조 방법 | KR1019820000725 | 1982-02-19 | KR1019830009124A | 1983-12-17 | 가주오구보-3 |
| 내용없음 | ||||||
| 74 | 생물학적 활성이 있는 헤테로 두고리형 히드록시미데이트와 타올리 히드록시미데이트 및 이들의 카르바메이트 에스테르 유도체 | KR1019810004271 | 1981-11-09 | KR1019830007701A | 1983-11-04 | 토마스에이매기외9 |
| 내용없음 | ||||||
| 75 | 電気導電性ポリマー組成物におけるジヘテロアミン | JP2018561988 | 2017-05-25 | JP6843889B2 | 2021-03-17 | ノラ サビナ ラドゥ; アルジャン ズームベルト |
| 76 | It substituted pyridoindole as agonists and antagonists of serotonin | JP2002559431 | 2001-12-19 | JP4231290B2 | 2009-02-25 | アルバート・ジェイ・ロビチョード; イアン・エス・ミッチェル; ウェンティン・チェン; ジョゼフ・カッチョラ; ジョン・エム・フェビッグ; テキュ・リー |
| 77 | 5ht2c receptor modulators | JP2006058747 | 2006-03-03 | JP4191741B2 | 2008-12-03 | スミス ジェフリー; スミス ブライアン |
| The present invention relates to novel compounds of formula (I): <CHEM> Which act as 5HT2C receptor modulators. These compounds are useful in pharmaceutical compositions whose use includes the treatment of obesity. <IMAGE> <IMAGE> <IMAGE> <IMAGE> <IMAGE> <IMAGE> <IMAGE> | ||||||
| 78 | 5ht2c receptor modulators | JP2003583332 | 2003-04-11 | JP4155926B2 | 2008-09-24 | ジェフリー スミス，; ブライアン スミス， |
| The present invention relates to novel compounds of formula (I): <CHEM> Which act as 5HT2C receptor modulators. These compounds are useful in pharmaceutical compositions whose use includes the treatment of obesity. <IMAGE> <IMAGE> <IMAGE> <IMAGE> <IMAGE> <IMAGE> <IMAGE> | ||||||
| 79 | Pyrrolo with atypical antipsychotic activity [2,1-b] de-alkylated derivatives of benzothiazepine | JP2007512730 | 2005-04-28 | JP2007536379A | 2007-12-13 | オルランド・ギラルディ; パオロ・カルミナティ; パトリツィア・ミネッティ; マリア・アッスンタ・ディ・チェサーレ; マリア・オルネーラ・ティンティ |
| 式(I)のピロロ[2,1-b]ベンゾチアゼピンの誘導体：式中、AはCH-CH
2 C=CH；Rは水素、ハロゲン、C
1 -C
4アルコキシ、C
1 -C
4アルキルチオ、C
1 -C
4アルキル、C
5 -C
6シクロアルキル；R
1は1-ピペラジニル、1-ホモピペラジニルおよび1-ピペリジニル；R
2は水素、C
1 -C
4アルコキシ、C
1 -C
4アルキルチオ、C
1 -C
4アルキル、CHO、CH=NOH、CH
2 OHである。 式(I)の化合物は特有の非定型の抗精神病活性を有し、それゆえ医薬、特に統合失調症、偏執症状態、躁鬱状態、情動領域の疾患、社会性の退行、人格の退行および幻覚の処置および予防のための医薬として有用である。 該化合物はまた有利な薬物動態学的特性を有する。
|
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| 80 | Useful new oxabispidine compounds in the treatment of cardiac arrhythmias | JP2001531792 | 2000-10-13 | JP3973906B2 | 2007-09-12 | ウィルスターマン，マイケル; クラディングボエル，デビッド; スヴェッソン，ペダー; ストランドルンド，ゲルト; トムソン，コリン; パヴェイ，ジョン; ブジェースン，マグヌス; ブジェレ，アンニカ; ホッフマン，クルト−ユルゲン; ポンテン，フリティオフ |
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