| 序号 | 专利名 | 申请号 | 申请日 | 公开（公告）号 | 公开（公告）日 | 发明人 |
|---|---|---|---|---|---|---|
| 101 | 트리아릴 유기보레이트의 제조 방법 | KR1020197016085 | 2017-11-07 | KR102489809B1 | 2023-01-20 | |
| 102 | 축합환 화합물 및 이를 포함한 유기 발광 소자 | KR1020190015192 | 2019-02-08 | KR1020200097870A | 2020-08-20 | |
| 103 | 미토플라보신: 플라빈-함유 효소를 표적화하여 미토콘드리아 호흡 억제에 의해 암 줄기 세포(CSCS)를 제거함 | KR1020207014732 | 2018-10-23 | KR1020200069365A | 2020-06-16 | |
| 104 | ２－ヨードソ安息香酸類の製造方法 | PCT/JP2019/049848 | 2019-12-19 | WO2020130081A1 | 2020-06-25 | 土肥 寿文; 知名 秀泰 |
本発明は高価な試薬を要せず、比較的安全に、ヨードソ安息香酸類を製造する方法の提供を目的とする。 本発明は、式（I）又は（II）：［式中、Arは、ベンゼン等を示し、R1、R21及びR22は、それぞれ独立して、ハロゲン等を示し、mは、nが0の場合は0-4の整数を、nが1の場合は0、1又は2を示し、nは0又は1を示し、r及びr'は、それぞれ独立して、0、1又を示す。］で表される化合物の製造方法であって式(III)又は(IV)： [式中、Q及びQ'は水素原子、アルカリ金属原子等を示し、x及びx'は2+又は+を示し、y及びzは1又は2を示し、Ar、R1、X、R21、R22、m及びnは前記と同じ。]で表される化合物を、水及び水と有機溶媒との混合溶媒から選択される溶媒中、ペルオキソ一硫酸モノカリウム及びオキソンから選択される少なくとも１つの過硫酸塩の存在下、0℃-100℃で酸化する工程を含む方法に関する。 |
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| 105 | DIAZOMETHYLATION REAGENT AND PROCESS FOR USING IT | PCT/EP2018/053190 | 2018-02-08 | WO2018146200A1 | 2018-08-16 | GARCÍA SUERO, Marcos; WANG, Zhaofeng |
The present invention relates compounds useful as reagents for the diazomethylation reaction, their preparation and the use thereof as reagents in a method for the diazomethylation reaction of aromatic substrates. It relates in particular to a compound of formula (I) wherein E is an electron withdrawing group. |
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| 106 | NOVEL IODINE COMPOUNDS, PROCESSES FOR THEIR PREPARATION AND USE THEREOF AS AMINATION AGENTS | PCT/EP2012/059638 | 2012-05-23 | WO2012160112A1 | 2012-11-29 | MUÑIZ KLEIN, Kilian; IGLESIAS GONZÁLEZ, Álvaro; SOUTO SALGADO, José Antonio; RÖBEN, Caren |
The iodine compounds of the present invention corresponds to those of formula (I), wherein R1, R1' and X have several meanings. These iodine compounds gives rise to the amination of several substrates without the need of catalysts, especially metal catalysts, and confer to the amination reaction the further advantage of being performed under mild conditions, which is of interest for industrial-scale production of nitrogenated compounds with pharmaceutical, biological or medicinal applications. Therefore, the iodine compounds of the invention are useful as amination agents. The invention also discloses several processes for the preparation of the iodine compounds of formula (I). |
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| 107 | SELECTIVE OXIDATION PROCESS WITH ENHANCED SAFETY | PCT/US0313070 | 2003-04-28 | WO03093210A8 | 2004-12-16 | CHIACCHIO UGO; RESCIFINA ANTONIO; MIRAGLIA GIUSEPPE; MAGNANO MARIANGELA; DI RAIMONDO PAOLA |
| A safe and effective process for the oxidation of a primary or secondary alcohol to the corresponding aldehyde or ketone via the reaction of said alcohol with an anhydride solution of a 1,1,1-tri(CZ-C4alkanoyloxy-1,1-dihydro-1,2-benziodoxol 3(1 H)-one, and a composition useful in this process. | ||||||
| 108 | METHOD FOR PRODUCING TRIARYLORGANOBORATES | US16950901 | 2020-11-17 | US20240002409A1 | 2024-01-04 | Thomas RÖLLE; Horst BERNETH; Dennis HÖNEL; Friedrich-Karl BRUDER; Jürgen KINTRUP |
| The invention relates to a process for preparing triaryl organo borates proceeding from organoboronic esters in the presence of an n-valent cation 1/n Kn+, comprising the anhydrous workup of the reaction mixture and the use of the triaryl organoborates obtained as co-initiator in photopolymer formulations, holographic media and holograms. | ||||||
| 109 | METHOD FOR PRODUCING TRIARYLORGANOBORATES | US16950906 | 2020-11-18 | US20220002321A1 | 2022-01-06 | Thomas RÖLLE; Horst BERNETH; Dennis HÖNEL; Friedrich-Karl BRUDER; Jürgen KINTRUP |
| The invention relates to a process for preparing triaryl organoborates proceeding from organoboronic esters in the presence of an n-valent cation 1/n Kn+, comprising the anhydrous workup of the reaction mixture and the use of the triaryl organoborates obtained as co-initiator in photopolymer formulations, holographic media and holograms. | ||||||
| 110 | Hypervalent iodine CF2CF2X reagents and their use | US16055629 | 2018-08-06 | US10669250B2 | 2020-06-02 | Vaclav Matousek; Petr Beier; Antonio Togni |
| Described herein are hypervalent iodine reagents. | ||||||
| 111 | IODONIUM ANALOGS AS INHIBITORS OF NADPH OXIDASES AND OTHER FLAVIN DEHYDROGENASES; FORMULATIONS THEREOF; AND USES THEREOF | US16160599 | 2018-10-15 | US20190048001A1 | 2019-02-14 | James Halpern DOROSHOW; Prabhakar RISBOOD; Jiamo LU; Krishnendu ROY; Charles T. KANE, JR.; Md Tafazzal HOSSAIN |
| Disclosed herein are novel iodonium analogs having anticancer and anti-inflammatory activity. | ||||||
| 112 | TRIFLUOROMETHOXYLATION OF ARENES VIA INTRAMOLECULAR TRIFLUOROMETHOXY GROUP MIGRATION | US16133297 | 2018-09-17 | US20190016670A1 | 2019-01-17 | Ming-Yu Ngai; Katarzyna N. Hojczyk |
| The present invention provides a process of producing a trifluoromethoxylated aryl or trifluoromethoxylated heteroaryl having the structure: wherein A is an aryl or heteroaryl, each with or without subsutitution; and R1 is —H, -(alkyl), -(alkenyl), -(alkynyl), -(aryl), -(heteroaryl), -(alkylaryl), -(alkylheteroaryl), —NH-(alkyl), —N(alkyl)2, —NH-(alkenyl), —NH-(alkynyl) —NH-(aryl), —NH-(heteroaryl), —O-(alkyl), —O-(alkenyl), —O-(alkynyl), —O-(aryl), —O-(heteroaryl); —S-(alkyl), —S-(alkenyl), —S-(alkynyl), —S-(aryl), or —S-(heteroaryl), comprising: (a) reacting a compound having the structure: with a trifluoromethylating agent in the presence of a base in a first suitable solvent under conditions to produce a compound having the structure: and (b) maintaining the compound produced in step (a) in a second suitable solvent under conditions sufficient to produce the trifluoromethoxylated aryl or trifluormethoxylated heteroaryl having the structure: | ||||||
| 113 | Iodonium analogs as inhibitors of NADPH oxidases and other flavin dehydrogenases; formulations thereof; and uses thereof | US15302566 | 2015-04-06 | US10131659B2 | 2018-11-20 | James Halpern Doroshow; Prabhakar Risbood; Jiamo Lu; Krishnendu Roy; Charles T. Kane, Jr.; Md Tafazzal Hossain |
| Disclosed herein are novel iodonium analogs having anticancer and anti-inflammatory activity. | ||||||
| 114 | Hypervalent iodine CF2CF2X reagents and their use | US15501872 | 2015-08-03 | US10040812B2 | 2018-08-07 | Vaclav Matousek; Petr Beier; Antonio Togni |
| A hypervalent iodine of formula (I) or formula (II) wherein R is a nucleophile and a method for their production is described. Such compounds can be used for fluoroethylation of compounds carrying a reactive group. A preferred compound carrying a reactive group is cystein in any environment such as peptide targets. | ||||||
| 115 | HYPERVALENT IODINE CF2CF2X REAGENTS AND THEIR USE | US15501872 | 2015-08-03 | US20170233420A1 | 2017-08-17 | Vaclav MATOUSEK; Petr BEIER; Antonio TOGNI |
| A hypervalent iodine of formula (I) or formula (II) wherein R is a nucleophile and a method for their production is described. Such compounds can be used for fluoroethylation of compounds carrying a reactive group. A preferred compound carrying a reactive group is cystein in any environment such as peptide targets. | ||||||
| 116 | Novel oxiodinium and thiaiodinium compounds | US337345 | 1973-03-02 | US4193935A | 1980-03-18 | William N. Cannon |
| Novel oxiodinium and thiaiodinium compounds having a superior inhibitory effect against micro-organisms coupled with outstanding stability and low toxicity are described. | ||||||
| 117 | Soluble salts of heterocyclic iodinecontaining bactericides | US44189065 | 1965-03-22 | US3332991A | 1967-07-25 | CANNON WILLIAM N |
| 118 | Process for inhibiting growth of microorganisms | US12344961 | 1961-07-12 | US3207660A | 1965-09-21 | CANNON WILLIAM N |
| 119 | A METHOD FOR FUNCTIONALIZATION OF AN AROMATIC AMINO ACID OR A NUCLEOBASE | EP20725768.4 | 2020-05-05 | EP3966203A1 | 2022-03-16 | MATOUSEK, Vaclav; BEIER, Petr; NOVAK, Petr |
| 120 | HYPERVALENT IODINE CF2CF2X REAGENTS AND THEIR USE | EP15750621.3 | 2015-08-03 | EP3180324B1 | 2020-11-25 | MATOUSEK, Václav; BEIER, Petr |
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