首页 / 专利分类库 / 有机化学 / 无环或碳环化合物 / 硫脲,即含下列基团NCSN或NCSN中的任何一个的化合物,其中的氮原子不属于硝基或亚硝基
序号 专利名 申请号 申请日 公开(公告)号 公开(公告)日 发明人
121 TR9802694 1997-06-24 TR199802694T2 1999-03-22 WIDDOWSON KATHERINE L
122 NO986110 1998-12-23 NO986110L 1999-02-23 WIDDOWSON KATHERINE L
123 Substituted benzenesulfonylureas and -thioureas, processes for their preparation and use of pharmaceutical preparations based on these compounds, and medicaments containing them AU4555996 1996-02-15 AU700254B2 1998-12-24 ENGLERT HEINRICH; GERLACH UWE; MANIA DIETER; GOEGELEIN HEINZ; KAISER JOACHIM
124 BENCENOSULFONILUREAS Y BENCENOSULFONILTIOUREAS SUSTITUIDAS, PROCEDIMIENTO PARA SU PREPARACION Y EMPLEO DE PREPARADOS FARMACEUTICOS A BASE DE ESTOSCOMPUESTOS, ASI COMO AGENTES CURATIVOS QUE LOS CONTIENEN. AR10139196 1996-02-15 AR002708A1 1998-04-29
La invención se refiere a bencenosulfonilureas y bencenosulfoniltioureas sustituidas de la fórmula (I) en donde R(1) es H, alquilo, cicloalquilo; R(2)es H, alquilo sustituido o nó con O, N, S, F, Cl, alcoxi, mercaptoalquilo, cicloalquilo; R(3) es H, alquilo sustituidos o nó por O, S, N, cicloalquilo,fluoralquilo, fluorocicloalquilo; R(4) es H, alquilo sustituido o nó con O, N, S, cicloalquilo, fluoroalquilo, fluorocicloalquilo ó R(3) y R(4) forman juntosun anillo de 2 a 8 miembros en elque uno o varios metilenos pueden estar reemplazados por heteroátomos; E es oxígeno o azufre; X es oxígeno o azufre; Yes [CR(5)R(5)]m: R(5) y R(5) son H o alquilo, m es un entero de 1 a 4, así como sus sales farmacéuticamente compatibles, que muestran extraordinariosefectos sobre el sistema cardiovascular.
125 Il-8 receptor antagonists AU3499497 1997-06-24 AU3499497A 1998-01-14 WIDDOWSON KATHERINE L
126 SUBSTITUTED BENZENESULFONYLUREAS AND -THIOUREAS, PROCESS FOR THEIR PREPARATION AND THE USE OF PHARMACEUTICAL PREPARATIONS BASED ON THESE COMPOUNDS, AS WELL AS MEDICAMENTS CONTAINING THEM HRP960076 1996-02-15 HRP960076A2 1997-12-31 KAISER JOACHIM
127 Substituted thiophenylsulfonylureas and -thioureas processes for their preparation their use as a medicament or diagnostic and medicament containing them ZA9600720 1996-01-31 ZA9600720B 1997-07-31 ENGLERT HEINRICH; HARTUNG JENS; CRAUSE PETER; MANIA DIETER; GOEGELEIN HEINZ; KAISER JOACHIM
N-((2-Benzamidoethyl)- thiophene-sulphonyl)-urea or-thiourea derivs. of formula (I) are new. R1 = H, halogen, Me, Et, OMe, OEt, SMe, SEt, 1-2C fluoroalkyl or 1-2C fluoroalkoxy; X = O or S; R2 = H, Me or CF3; Y, Z = H, F, Cl, Br, I, Me, Et, OMe or OEt.
128 Process for the vacylation of threonine derivatives and their use in the preparation of 1,4-dihydropyridines. GR970400402 1997-03-03 GR3022713T3 1997-06-30 STOLTEFUSS JUERGEN DIPL-ING; BECHEM MARTIN DR; GROSS RAINER PROF DR; HEBISCH SIEGBERT DR; SCHRAMM MATTHIAS DR
129 AT89110528 1989-06-10 ATE149154T1 1997-03-15 STOLTEFUSS JUERGEN DI; BECHEM MARTIN DR; GROSS RAINER PROF-DR; HEBISCH SIEGBERT DR; SCHRAMM MATTHIAS DR
130 A process for the acylation of threonine derivatives and their use for the preparation of 1,4-dihydropyridines DE58909770 1989-06-10 DE58909770D1 1997-03-06 STOLTEFUSS JUERGEN DIPL ING; BECHEM MARTIN DR; GROSS RAINER PROF DR; HEBISCH SIEGBERT DR; SCHRAMM MATTHIAS DR
131 SUBSTITUTED TIOPHENSULFONYL UREAS AND THIOUREAS, PROCESS FOR THE PREPARATION THEREOF, USE THEREOF AS MEDICINE OR AS DIAGNOSTIC AS WELL AS MEDICINE CONTAINING THEM SI9600033 1996-02-01 SI9600033A 1996-10-31 ENGLERT HEINRICH; HARTUNG JENS; CRAUSE PETER; MANIA DIETER; GOEGELEIN HEINZ; KAISER JOACHIM
132 N-(AMINO(THIO)CARBONYLALKYL)BENZENESULPHONYL (THIO)UREA DERIVATIVES NZ28099296 1996-02-15 NZ280992A 1996-10-28 ENGLERT HEINRICH; GERLACH UWE; MANIA DIETER; GOEGELEIN HEINZ; KAISER JOACHIM
133 N-[2-(BENZOYLAMINOETHYL)THIENYLSULPHONYL](THIO)UREA DERIVATIVES NZ28089096 1996-01-26 NZ280890A 1996-10-28 ENGLERT HEINRICH; HARTUNG JENS; CRAUSE PETER; MANIA DIETER; GOGELEIN HEINZ; KAISER JOACHIM
134 SUBSTITUTED BENZENESULFONYLUREAS AND -THIOUREAS, METHOD OF THEIR MANUFACTURE AND APPLICATION OF PHARMACEUTICALS ON BASE OF THESE COMPOUNDS AND MEDICAMENTS CONTAINING THEM SK21296 1996-02-15 SK21296A3 1996-10-02 ENGLERT HEINRICH; GERLACH UWE; MANIA DIETER; GOEGELEIN HEINZ; KAISER JOACHIM
Substituted benzene sulphonyl urea and thiourea compounds of formula (I), wherein R(1), R(2), R(3), R(4), E, X and Y has the meaning given in claims. The said compounds are effective for cardiovascular system.
135 СПОСОБ ПОЛУЧЕНИЯ 2-АМИДИНОТИОМОЧЕВИНЫ SU3277065 1981-01-09 SU1091512A1 1996-09-20 TOMCHIN A B; STOPSKIJ V S
1. Способполучения 2-амидинотиомочевиныс использованиемдициандиамида, отличающийсятем, что, сцельюупрощенияпроцесса, дициандиамидподвергаютвзаимодействиюс гидросульфидомаммонияприрН 7,8 - 9,6 притемпературе 35 - 90С.2. Способпоп. 1, отличающийсятем, чтоиспользуютгидросульфидаммония, полученныйнепосредственнов реакционнойсреде.
136 SUBSTITUTED BENZENESULFONYL UREAS AND BENZENESULFONYLTHIOUREAS, PROCESS OF THEIR PREPARATION AND USE OF PHARMACEUTICAL PREPARATIONS BASED ON SAID COMPOUNDS, AS WELL AS MEDICAMENTS CONTAINING THEREOF CZ43596 1996-02-14 CZ43596A3 1996-09-11 ENGLERT HEINRICH; GERLACH UWE; MANIA DIETER; GOEGELEIN HEINZ; KAISER JOACHIM
137 NO960628 1996-02-16 NO960628L 1996-08-19 ENGLERT HEINRICH; GERLACH UWE; MANIA DIETER; GOEGELEIN HEINZ; KAISER JOACHIM
138 Substituted Thiophenylsulfonylharnstoffe and thioureas, processes for their preparation, their use as a medicament or diagnostic, and drug containing them DE19503136 1995-02-01 DE19503136A1 1996-08-08 ENGLERT HEINRICH CHRISTIAN DR; HARTUNG JENS DR; CRAUSE PETER DR; MANIA DIETER DR; GOEGELEIN HEINZ DR; KAISER JOACHIM DR
139 NO960411 1996-01-31 NO960411L 1996-08-02 ENGLERT HEINRICH; HARTUNG JENS; CRAUSE PETER; MANIA DIETER; GOGELEIN HEINZ; KAISER JOACHIM
140 Substituted benzenesulfonylureas and -thioureas processes for their preparation and use of pharmaceutical preparation based on these compounds and medicaments containing them IL11715296 1996-02-15 IL117152D0 1996-06-18
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