序号 专利名 申请号 申请日 公开(公告)号 公开(公告)日 发明人
141 JPS59501982A - JP50301083 1983-09-23 JPS59501982A 1984-11-29
142 Plant growth regulator JP2968884 1984-02-21 JPS59157067A 1984-09-06 HANSU GEORUKU SHIYUMITSUTO; KURAUSU RIYURUSEN; KARURUFURIITO BEDEMAIYAA
143 Diffusion transfer photographic film unit JP25247083 1983-12-28 JPS59136732A 1984-08-06 ABINATSUSHIYU SHII META
144 Propionic acid derivative and manufacture JP24235483 1983-12-23 JPS59130236A 1984-07-26 SEIKE KOUICHI; UBE PURIISUNITSUTSU; HANSUUYOTSUHEMU RIIBERU; RUUTOUITSUHI OIE; ROBERUTO AARU SHIYUMITSUTO
145 Enantiomer of propionic acid derivative and manufacture JP24235383 1983-12-23 JPS59130235A 1984-07-26 SEIKE KOUICHI; UBE PURIISUNITSUTSU; HANSUUYOTSUHEMU RIIBERU; RUUTOUITSUHI OIE; ROBERUTO AARU SHIYUMITSUTO
146 Leucotriene antagonist JP18099883 1983-09-30 JPS5993043A 1984-05-29 PATORISU SHII BERANJIYAA; REJIYAN FUOOTEIN; IBUAN GIYUINDON; JIYOSHIYUA ROKATSUCHI; KURISUCHIYAN YOAKIMU
147 Benzhydrylsulfinylacetamide derivative, manufacture and central nervous system therapy JP9879883 1983-06-04 JPS591459A 1984-01-06 RUI RAFUON
148 Polyanionic compound, manufacture and composition JP1728983 1983-02-04 JPS58145795A 1983-08-30 GIYUI BANRERUBERUGE; ANRI SEBATSUGU
149 Manufacture of alpha,alpha-difluoroalkoxy or alpha,alpha-difluoroalkylthiophenylsulfone JP11088082 1982-06-29 JPS58124760A 1983-07-25 MISHIERU DEBOWA
150 Aminophenol derivative, its preparation and remedy containing the same JP20974081 1981-12-28 JPS58113152A 1983-07-05 WAKATSUKA HIROHISA; MOURI TETSUYA; HASHIMOTO SHINSUKE
NEW MATERIAL:A compound of formulaI[R is formula II(Z is thio, sulfinyl; n is 1, 2, 3; R 1 is H, alkyl, halogen, hydroxyl), formula III (R 2 is H, alkyl, halogen; m is 1, 2), formula IV and formula V]. EXAMPLE: 2-Amino-4-phenylthiophenol. USE: A preventive of or remedy for allergic tracheitis, bronchitis, pneumonopathy, a variety of inflammations and a variety of inflammation caused by prostaglandins. PREPARATION: The selective reduction of the nitro group in the 2-position of the compound of formulaIis conducted with a hydrogen gas in the presence of a catalyst such as Ni, Pt or Pd on carbon or by using Fe, Zn, Sn or SnCl 2 and hydrochloric acid to give the compound of formulaIwith NH 2 group. COPYRIGHT: (C)1983,JPO&Japio
151 JPS5757015B2 - JP13975878 1978-11-13 JPS5757015B2 1982-12-02 TOOMASU HENRII ORUZAISU; CHAARUZU AAMON HAABAATO; MAIKERU ROSU JONSON; ROORENSU SHAAMAN MERUBIN JUNIAA
Compounds of the formula <IMAGE> <IMAGE> wherein R1 is hydrogen, benzyl, benzoyl, alkanoyl of 1 to 5 carbon atoms or -CO-(CH2)p-NR'R'' wherein p is 0 or an integer from 1 to 4; each of R' and R'' when taken individually is hydrogen or alkyl of 1 to 4 carbon atoms; R' and R'' when taken together with the nitrogen to which they are attached form a 5- or 6-membered heterocyclic ring selected from piperidino, pyrollo, pyrrolidino, morpholino and N-alkylpiperazino having from 1 to 4 carbon atoms in the alkyl group; R2 is selected from hydrogen, alkanoyl of 1 to 6 carbon atoms and benzoyl; R3 is selected from hydrogen, methyl and ethyl; R4 is selected from hydrogen, alkyl of 1 to 6 carbon atoms and benzyl; Z is selected from: (a) alkylene having from one to nine carbon atoms; (b) -(alk1)m-X-(alk2)n- wherein each of (alk1) and (alk2) is alkylene having from 1 to 9 carbon atoms, with the proviso that the summation of carbon atoms in (alk1) plus (alk2) is not greater than 9; m and n are each 0 or 1; X is selected from O, S, SO, and SO2; and W is selected from hydrogen, methyl, pyridyl, piperidyl, phenyl, monochlorophenyl, monofluorophenyl and <IMAGE> wherein W1 is selected from hydrogen, phenyl, monochlorophenyl and monofluorophenyl; a is an integer from 1 to 5 and b is 0 or an integer from 1 to 4, with the proviso that the sum of a and b is not greater than 5. Compounds I and II are useful as analgesics. Compound III is useful as an intermediate for the preparation of Compounds I and II. Intermediates for the preparation of I, II and III are disclosed. A process for the use of compounds I and II to produce analgesia is also described.
152 Salt of 5-fluoro-2-methyl-1-(p- (methylsulfinyl)benzylidene)indene-3-acetic acid JP4703282 1982-03-23 JPS57167958A 1982-10-16 KARURO MIRANI; JIOBANNI MARIA KARUMINAACHI; ATSUCHIRIO SOBEERA
153 JPS5736899B2 - JP1823977 1977-02-23 JPS5736899B2 1982-08-06
154 JPS5727107B1 - JP10151170 1970-11-19 JPS5727107B1 1982-06-08
155 4-substituted 3,3-dimethyl-butane-2-ones and manufacture JP8583581 1981-06-05 JPS5726636A 1982-02-12 BUORUFUGANGU KUREEMAA; HANSUURUUTOUITSUHI ERUBE
156 JPS5640152B2 - JP14229777 1977-11-29 JPS5640152B2 1981-09-18
157 JPS5640151B1 - JP769372 1972-01-21 JPS5640151B1 1981-09-18
158 JPS5639281B2 - JP11037475 1975-09-11 JPS5639281B2 1981-09-11
159 JPS5638587B1 - JP630078 1978-01-25 JPS5638587B1 1981-09-08
160 JPS5636163B2 - JP9076074 1974-08-09 JPS5636163B2 1981-08-22
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