子分类：
| 序号 | 专利名 | 申请号 | 申请日 | 公开（公告）号 | 公开（公告）日 | 发明人 |
|---|---|---|---|---|---|---|
| 21 | Coupling of nucleophiles, vinyl compounds or CO with water, alcohols or amines to organic compounds | US09799084 | 2001-03-06 | US20010037042A1 | 2001-11-01 | Adriano Indolese; Anita Schnyder |
| Process for the coupling of a) nucleophiles selected from the group alcohols, thioles, amines, metallised hydrocarbons, CH-acidic compounds and metal cyanides, or of b) carbon monoxide mixed with water, alcohols, ammonia, primary or secondary amines, to organic compounds selected from the group of leaving-group-containing aromatics, hetero-aromatics with a C-bonded leaving group, aromatic or hetero-aromatic methyl compounds with a leaving group bonded to the methyl group, ethylenically unsaturated organic compounds with a C-bonded leaving group, or organic allyl compounds with a leaving group in allyl position, or c) vinyl compounds with leaving-group-containing aromatics, whilst cleaving the leaving group in the presence of Pd complexes with monophospholine ligands as the catalyst, whereby variants b) and c) are carried out in the presence of an inorganic base or organic nitrogen base, the process being characterised in that the Pd complex contains secondary monophosphines with aliphatic, branched or cyclic substituents as ligands. | ||||||
| 22 | Bisphenol ester derivatives | US562774 | 1995-11-27 | US5602196A | 1997-02-11 | Bernard Gilg; Rita Pitteloud |
| Stabilisers of formula I ##STR1## wherein R.sub.1 and R.sub.2 may be C.sub.1 -C.sub.5 alkyl, the substituents R.sub.3 to R.sub.8 may be hydrogen, the variable n may be 1 or 2, and, when n is 1, A may be an alkoxy radical, and, when n is 2, A may be a diamine radical. | ||||||
| 23 | Soft tertiary amine esters of bio-affecting carboxylic acids | US202750 | 1980-10-31 | US4381307A | 1983-04-26 | Kenneth B. Sloan |
| Novel derivatives of known bio-affecting carboxylic acids R-COOH are disclosed, said derivatives having the structural formula ##STR1## wherein Y and Y' are each H or C.sub.1 -C.sub.4 alkyl; n is 0 or 1; R.sub.1 and R.sub.2 are each selected from a variety of unsubstituted or substituted hydrocarbon radicals, or are combined so that --NR.sub.1 R.sub.2 represents the residue of a saturated or unsaturated heterocyclic compound containing one secondary nitrogen atom; and R.sub.3 is H or one of a variety of other substituents. Salts and N-oxides of compounds of formula (I) and the corresponding diacyloxy derivatives of known bio-affecting carboxylic acids HOOC-R'-COOH are disclosed also. The parent acids from which the subject soft tertiary amine esters can be derived include such bio-affecting agents as cephalosporin and penicillin antibiotics, amino acids and structurally related compounds, prostaglandins and their metabolites, steroidal anti-inflammatory agents, and non-steroidal anti-inflammatory/non-narcotic analgesic/antipyretic agents. | ||||||
| 24 | (메타)아크릴레이트계 화합물, 이를 포함하는 감광성 수지 조성물 및 이미지 센서 | KR1020090046036 | 2009-05-26 | KR101266298B1 | 2013-05-22 | 정의준; 이창민; 김재현; 이길성; 샤로크몰탈베비; 시나마그수디 |
| 본명세서에서는에스테르산소를갖는 (메타)아크릴레이트기적색광을생성하는투과스펙트럼을갖는치환또는비치환된안트라퀴논기및 상기 (메타)아크릴레이트기의에스테르산소및 치환또는비치환된안트라퀴논기와공유결합하는연결기를포함하고, 상기연결기는치환또는비치환된탄소수 3 내지 10의알킬렌기, 치환또는비치환된탄소수 3 내지 20의사이클로알킬렌기및 치환또는비치환된탄소수 6 내지 30의아릴렌기로이루어진군으로부터선택되는기를포함하는것인 (메타)아크릴레이트계화합물, 이를포함하는감광성수지조성물및 이미지센서가제공된다. | ||||||
| 25 | Process for the production of triaryl organoborates | US16348262 | 2017-11-07 | US11078218B2 | 2021-08-03 | Thomas Rölle; Horst Berneth; Dennis Hönel; Friedrich-Karl Bruder |
| Provided herein is a process for preparing triaryl organoborates proceeding from alkyl or cycloalkyl boronates in the presence of an n-valent cation 1/n Kn+ to obtain organoborates of the formula 1/n Kn+R34B−—R1 (IV), where one equivalent of organoboronic ester of the formula B—R1(OR2)(OR3) (I) is initially charged together with 1/n equivalents of salt Kn+ nX− (II) and 3 equivalents of metal M in a solvent or a solvent mixture, 3 equivalents of a haloaromatic R4—Y (III) are added, and optionally a second organic solvent water is added and the compound 1/n Kn+ R24B−—R1 (IV) is separated off with the organic phase, and to the use of these substances as co-initiator in photopolymer formulations. | ||||||
| 26 | Biodegradable poly (phosphoester-co-desaminotyrosyl L-tyrosine ester) compounds, compositions, articles and methods for making and using the same | US834164 | 1997-04-14 | US5912225A | 1999-06-15 | Hai-quan Mao; Kam W. Leong |
| Biodegradable polymers are described comprising the recurring monomeric units shown in formula I: ##STR1## wherein: R is selected from the group consisting of H, alkyl, aryl or heterocyclic; andR' is selected from the group consisting of H, alkyl, alkoxy, aryl, aryloxy, heterocyclic or heterocycloxy; andn is 5 to 500,wherein said biodegradable polymer is biocompatible before and upon biodegradation.Processes for preparing the polymers, compositions containing the polymers and biologically active substances, articles useful for implantation or injection into the body fabricated from the compositions, and methods for controllably releasing biologically active substances using the polymers, are also described. | ||||||
| 27 | Quaternized esters | US949260 | 1992-11-16 | US5296622A | 1994-03-22 | Guenter Uphues; Uwe Ploog; Rainer Jeschke; Peter Waltenberger |
| Quaternized esters having fabric-softening and hydrophilicizing properties are obtained by reaction of unsaturated fatty acids containing at least 40 mol-% transconfigured double bonds or esters thereof with alkanolamines and subsequent quaternization of the reaction products with alkylating agents. | ||||||
| 28 | Organic quaternary ammonium compounds and process for the preparation thereof | US807785 | 1985-12-11 | US4675131A | 1987-06-23 | Rene Walraevens; Jean-Marc Coisne |
| Quaternary ammonium compounds having the general formula: ##STR1## in which, R.sub.1 is an alkyl or aryl group, unsubstituted or substituted by at least two ester groups;R.sub.2, R.sub.3 and R.sub.4 are alkyl, aryl, aryl alkyl or alkyl aryl groups substituted by ester groups comprising no more than 10 carbon atoms;m, r and n are whole numbers;A.sup. .circle.r- is an anion such that m.times.r=n. The compounds are obtained by treatment of a tert.alcohol-amine with an alkylating or arylating agent and an acylating agent. They may be used as activators of persalts in wash compositions. | ||||||
| 29 | Biodegradable zwitterionic surfactant compounds | US114184 | 1980-01-22 | US4301044A | 1981-11-17 | George E. Wentler; Joseph McGrady; Eugene P. Gosselink; William A. Cilley |
| Zwitterionic surfactant compounds are made readily biodegradable in the environment by the inclusion of a biochemically and/or hydrolytically labile chemical linkage located between the cationic and anionic charge centers of the compounds and anywhere from the second to the tenth atom distant from the cationic charge center. The biodegradable linkage is preferably an ester or amide. The alkoxylated zwitterionic surfactants herein exhibit outstanding particulate soil removal performance and are also effective in removing oily soils from fabrics, in addition to being readily biodegradable. Also described are detergent compositions containing the zwitterionic surfactants, and, optionally containing cosurfactants and detergent builders. | ||||||
| 30 | Novel fatty acid derivatives | JP53186398 | 1998-01-23 | JP4698773B2 | 2011-06-08 | サンドボルド、マリット・リラント; ダレン、アレ; ビョレッツェン、ベルント; マイレン、フィン |
| 31 | Pharmaceutical compounds | JP2001516885 | 2000-07-27 | JP2003515526A | 2003-05-07 | ソルダト，ピエロ デル |
| (57)【要約】 一般式(Ｉ）の化合物またはその塩：Ａ−Ｂ−Ｎ(Ｏ) S ［式中、ｓは１または２に等しい整数であり；Ａ＝Ｒ−Ｔ 1 -であり 、ここで、Ｒは薬物の残基であり、Ｔ 1 ＝(ＣＯ) tまたは(Ｘ) t'であり、ここで、Ｘ＝Ｏ、Ｓ、ＮＲ 1Cであり、Ｒ 1CはＨまたは直鎖状または分枝鎖状のアルキルまたは遊離原子価であり、ｔおよびｔ'は、ｔ'＝０のときｔ＝１であり、ｔ'＝１のときｔ＝０であるという条件付きで、０または１に等しい整数であり；Ｂ＝-Ｔ B −Ｘ 2 −Ｏ-であり、ここで、ｔ＝０のときＴ B ＝(ＣＯ)であり、ｔ'＝０のときＴ B ＝Ｘであり、Ｘは上記で定義されたとおりであり；二価の基Ｘ 2は、Ａの前駆薬物およびＢの前駆体が、明細書に記載の薬理試験にそれぞれ適合するようなものである。 | ||||||
| 32 | The novel tetrahydronaphthalene compounds prepared by the rhodium-catalyzed ring-opening reaction in the presence of a phosphine ligand | JP2001533091 | 2000-10-26 | JP2003512446A | 2003-04-02 | キース・ファグヌー; マーク・ラウテンス |
| (57)【要約】 本発明は、ヒドロナフタレン環構造を有するエナンチオマー的に富んだ化合物の製造方法に向けられる。 この方法は、ロジウムを触媒として用い、そしてホスフィン配位子の存在下に、オキサベンゾノルボルナジエンを求核試薬と反応させることを伴う。 合成される化合物は種々の疾患および状態を処置するための医薬調製物に使用できる。 | ||||||
| 33 | Optically active alcohol and carboxylic acid ester thereof | JP35242396 | 1996-12-13 | JPH10175926A | 1998-06-30 | ABIKO ATSUSHI; RIYUU KEIHOU |
| PROBLEM TO BE SOLVED: To obtain the subject new compound having an α-H and useful for the synthesis of an optically active anti-aldol by enolizing in the presence of boron triflate and an amine, and then reacting with an aldehyde. SOLUTION: This optically active alcohol is a new compound expressed by formula I (R<1> to R<6> are each H, an alkyl, etc.), e.g. 2-(N-methylenesulfonyl) amino-1-phenyl-1-propanol. The method for producing the compound of formula I is constituted by e.g. using norephedrine as a raw material, performing an N-sulfonylation reaction of the raw material by mesitylene sulfonylchloride and (C2 H5 )3 N in CH2 Cl2 to form a compound of formula II, then performing an N-benzylation reaction of the above compound with benzyl bromide and K2 CO3 in CH3 CN to form an optically active alcohol of formula III, and esterifying the alcohol with propionyl chloride and pyridine in CH2 Cl2 to form a carboxylic acid ester expressed by formula IV. | ||||||
| 34 | JPS6254298B2 - | JP9939079 | 1979-08-03 | JPS6254298B2 | 1987-11-13 | EDOWAADO ROTSUKUTSUDO UIIRAA; ERUMAA HARII JANSHISU; RICHAADO ANSONII JENKARERI; FURANKURIN HAABAATO BAROZU |
| 35 | Organic quaternary ammonium compound | JP28016185 | 1985-12-12 | JPS61180747A | 1986-08-13 | RUNE WARURABENZU; JIYAN MARUKU KOWASUNU |
| 36 | JPS6129348B2 - | JP9939179 | 1979-08-03 | JPS6129348B2 | 1986-07-05 | EDOWAADO ROTSUKUTSUDO UIRAA; ERUMAA HARII JANSHISU; RICHAADO ANSONII JENKARERI; FURANKURIN HAABAATO BAROZU |
| 37 | Vitally influencing soft tertiary amine ester of carboxylic acid | JP17373881 | 1981-10-31 | JPS57106647A | 1982-07-02 | KENESU BII SUROON |
| 38 | Biodegradable zwitterionic surfactant compound and detergent composition containing it | JP854281 | 1981-01-22 | JPS56150048A | 1981-11-20 | JIYOOJI EDOWAADO UENTORAA; JIYOSEFU MAKUGURADEII; YUUJIN POORU GOSERINKU; UIRIAMU AJIARON SHIRII |
| 39 | New fatty acid derivative | JP2009141714 | 2009-06-12 | JP2009280583A | 2009-12-03 | MYHREN FINN; DALEN ARE; BORRETZEN BERNT; SANDVOLD MARIT LILAND |
| <P>PROBLEM TO BE SOLVED: To provide a method for improving the actions of many biologically active compounds such as drugs and agrochemicals by a chemical derivatization method. <P>SOLUTION: The properties of biologically active compounds such as drugs and agrochemicals containing in their molecular structure one or more functional groups selected from an alcohol, ether, phenyl, amino, amide, thiol, carboxylic acid and carboxylic acid ester groups are modified by replacing one or more of these functional groups by a lipophilic group selected from those of formula: RCOO-, RCONH-, RCOS-, RCH<SB>2</SB>O-, RCH<SB>2</SB>NH-, -COOCH<SB>2</SB>R and -SCH<SB>2</SB>R, wherein R is a lipophilic moiety selected from cis-8-heptadecenyl, trans-8-heptadecenyl, cis-10-nonadecenyl and trans-10-nonadecenyl. <P>COPYRIGHT: (C)2010,JPO&INPIT | ||||||
| 40 | Optically active alcohol and the carboxylic acid ester | JP35242396 | 1996-12-13 | JP3770678B2 | 2006-04-26 | 継峰 劉; 淳 安孫子 |
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