序号 专利名 申请号 申请日 公开(公告)号 公开(公告)日 发明人
341 A combination of heat stabilizer / lubricant for PVC processing and method for their preparation DE69425089 1994-01-27 DE69425089D1 2000-08-10 BEEKMAN GEORGE F; MESCH KEITH A; PRICE LIONEL R
342 AT94300619 1994-01-27 ATE194368T1 2000-07-15 BEEKMAN GEORGE F; MESCH KEITH A; PRICE LIONEL R
343 AT95944790 1995-10-25 ATE194337T1 2000-07-15 DELORME DANIEL; DUCHARME YVES; FRIESEN RICHARD; GRIMM ERICH L; LEPINE CAROLE
344 ACETIC ACID DERIVATIVES RU94042929 1994-12-02 RU2151768C1 2000-06-27 ALIG LEO; KHADVARI POL; KHJURTSELER MJULLER MARIANNE; MJULLER MARSEL; SHTAJNER BEAT; VELLER TOMAS
chemical industry. SUBSTANCE: described are acetic acid derivatives of formula I: wherein L, M, Q and T are as defined in claim 1. Compounds are useful for treatment or prophylaxis of diseases associated with binding of adhesive proteins with thrombicytes and also aggregation of thrombicytes and cell-cell adhesion. Compounds are prepared by detachment of protective groups in corresponding protected compounds or by conversion of cyan group into amidine group in corresponding nitriles. EFFECT: improved properties of the title compounds. 23 cl, 193 ex, 1 tbl
345 Acetic acid derivatives as drugs DE59409322 1994-11-26 DE59409322D1 2000-06-08 ALIG LEO; HADVARY PAUL; HUERZELER MUELLER MARIANNE; MUELLER MARCEL; STEINER BEAT; WELLER THOMAS
346 Brefeldin and analogs for enhanced synaptic transmission DK95930845 1995-08-16 DK0782573T3 2000-06-05 SUMIKAWA KATUMI; ITO KEN-ICHI; MCGAUGH JAMES L
347 4,5-disubstituted 2-phenylphenol leukotriene antagonists and pharmaceutical compositions containing them IL10384792 1992-11-23 IL103847A 2000-06-01
348 PT96402423 1996-11-13 PT776881E 2000-05-31 BERNARDON JEAN-MICHEL; CHARPENTIER BRUNO
349 Bi-aromatic compounds comprising an adamantyl group in para-position, pharmaceutical and cosmetic compositions containing them and their utilization GR20000400316 2000-02-09 GR3032617T3 2000-05-31 BERNARDON JEAN-MICHEL; CHARPENTIER BRUNO
350 Biaromatic compounds having adamantyl group in the para-position, pharmaceutical and cosmetic compositions containing them, and uses DE69605525 1996-11-13 DE69605525T2 2000-05-04 BERNARDON JEAN-MICHEL; CHARPENTIER BRUNO
351 Diaromatiske compounds bearing an adamantyl group in the para position, pharmaceutical and cosmetic preparations which incorp DK96402423 1996-11-13 DK0776881T3 2000-04-25 BERNARDON JEAN-MICHEL; CHARPENTIER BRUNO
352 Derivatives of 2-cyano-1-sulfonamidophenyl-1,3-dione and their use as herbicides. ES97109375 1994-05-13 ES2141559T3 2000-03-16 CRAMP SUSAN MARY; PETTIT SIMON NEIL; MUSIL TIBOR; SMITH PHILIP HENRY GAUNT
LA INVENCION SE REFIERE A DERIVADOS 2 NA DE FORMULA: EN LA QUE R, R{SUP,1}, R{SUP,2}, R{SUP,3}, R{SUP,4} YR{SUP,5} SE DEFINEN EN LA DESCRIPCION, CON LA CONDICION DE QUE AL MENOS UNO DE LOS GRUPOS R{SUP,2} AR{SUP,5} REPRESENTA N(R{SUP,12})SO{SUB,2}R{SUP,8}; DONDE R{SUP,8} YR{SUP,12} SON COMO SE DEFINE EN LA DESCRIPCION, Y SU USO COMO HERBICIDAS.
353 CARBAMOYLCARBOXILIC ACID AMIDES, METHOD OF PREPARATION THEREOF, AGENT AND METHODS FOR CONTROLLING PATHOGENOUS FUNGI RU97105197 1995-08-19 RU2145956C1 2000-02-27 FRANK VETTERIKH; OLIVER VAGNER; KARL AJKKEN; EHBERKHARD AMMERMANN; GIZELA LORENTS
FIELD: biologically- active compounds. SUBSTANCE: invention provides new carbamoylcarboxilic acid amides with general formula I: (I), wherein R1 is C1-C8-alkyl, R2 hydrogen, R3 C1-C8-alkyl, R4 and R5 are hydrogen atoms, X, independently, are hydrogen or C1-C8-alkyl, Y, independently, are one of X radicals, q and p, independently, are 0 or 1, provided that they cannot simultaneously be equal to 0, and r is 0, 1, or 2, and salts of these compounds showing fungicidal activity. EFFECT: extended choice of fungicides. 7 cl, 5 tbl
354 Substituted cyclopentylaminderivate and antagonists whose use as a calcium-channel DE69510192 1995-03-14 DE69510192T2 2000-02-24 BROWN THOMAS; HARLING JOHN; ORLEK BARRY
355 AT97109375 1994-05-13 ATE189212T1 2000-02-15 CRAMP SUSAN MARY; PETTIT SIMON NEIL; MUSIL TIBOR; SMITH PHILIP HENRY GAUNT
356 (3S- (3R*, 4aR*, 8aR*, 2'S*, 3'*))-2-(2'-hydroxy-3'-phenylthiomethyl (or benzyl, napthylthiomethyl, or methylnaphthyl)-4'-aza-5'-oxo-5'-(2"-methyl-3"-hydroxyphenyl) pentyl) decahydroisoquinoline-3-N-t-butylcarboxamide and its pharmaceutically acceptable salts and its prodrug analogs IL12509894 1994-10-31 IL125098A 2000-01-31
357 Bio-aromatic, containing an adamantyl group in the para-position of compounds containing these pharmaceutical and cosmetic compositions and their use DE69605525 1996-11-13 DE69605525D1 2000-01-13 BERNARDON JEAN-MICHEL; CHARPENTIER BRUNO
358 amine acids method for synthesis of alpha-substituted Akrylsäuren and N- (mercaptoacyl) DE69603101 1996-03-01 DE69603101T2 1999-12-09 DUHAMEL PIERRE; DUHAMEL LUCETTE; DANVY DENIS; MONTEIL THIERRY; LECOMTE JEANNE-MARIE; SCHWARTZ JEAN-CHARLES
359 NO963030 1996-07-19 NO306396B1 1999-11-01 BECKETT RAYMOND PAUL; WHITTAKER MARK; MILLER ANDREW; MARTIN FIONNA MITCHELL
360 ACETIC ACID DERIVATIVES, METHODS FOR THEIR PREPARATION AND APPLICATION BG9923394 1994-12-02 BG62399B1 1999-10-29 ALIG LEO; HADVARY PAUL; HUERZELER MUELLER MARIANNE; MUELLER MARCEL; STEINER BEAT; WELLER THOMAS
The derivatives are used for the treatment or prevention ofdiseases caused by binding of adhesive proteins and thrombocytesfrom the trombocydal aggregation and intercellular adhesion. Theyhave the formulawhere radicals L, M, Q & T have the meanings listed in thedescription. They are produced by splitting of the protectiongroups into the respective protected compounds or by theconversion of the cyanogroup of the respective mitriles into anamidinogroup.25 claims
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