序号 | 专利名 | 申请号 | 申请日 | 公开(公告)号 | 公开(公告)日 | 发明人 |
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41 | Insecticide mainly composed of selected neonicotinoids and strobilurins | JP2011256488 | 2011-11-24 | JP2012087134A | 2012-05-10 | KROHN PETER-WILHELM; BECKER ROLF CHRISTIAN; HUNGENBERG HEIKE |
PROBLEM TO BE SOLVED: To provide a composition having excellent insecticidal property and bactericidal property.SOLUTION: There are provided pesticides for plants, using a composition comprising an active material selected from neonicotinoids (clothianidin, imidacloprid, thiacloprid, dinotefuran, acetamiprid, nitenpyram, and thiamethoxam) and at least one active material selected from strobilurin bactericides (picoxystrobin, pyraclostrobin, dimoxystrobin, metominostrobin and orysastrobin). These can be used as a dust coating agent of seed, for seed treatment. | ||||||
42 | Production of dideoxynucleoside derivative by selective hydrolysis | JP33195289 | 1989-12-21 | JPH03190876A | 1991-08-20 | SHIRAGAMI HIROSHI; TANAKA YASUHIRO; IWAGAMI TOSHIO |
PURPOSE: To easily and selectively obtain the subject compound useful as pharmaceuticals on an industrial scale at a low cost by hydrolyzing a specific nucleoside compound in a solution in the presence of a cyclodextrin and an inorganic salt and subjecting the product to hydrogenation reaction. CONSTITUTION: The objective compound of formula V (R 3 is 1-12C hydrolyzable acyl or H) can be produced by hydrolyzing a compound of formula I (B is nucleic acid base; R 1 and R 2 are 1-12C hydrolyzable acryl; X is H, halogen, 1-12C alkyl, etc.) or formula II in a solution in the presence of a cyclodextrin and an inorganic salt, converting the hydroxyl group of the resultant compound of formula III or formula IV to another substituent having high eliminability, hydrogenating the product and, as necessary, further hydrolyzing the reaction product. COPYRIGHT: (C)1991,JPO&Japio | ||||||
43 | SELEKTIVE INSEKTIZIDE UND/ODER AKARIZIDE AUF BASIS VON SUBSTITUIERTEN, CYCLISCHEN DICARBONYLVERBINDUNGEN UND SAFENERN | PCT/EP2005/007790 | 2005-07-18 | WO2006008107A1 | 2006-01-26 | FISCHER, Reiner; RECKMANN, Udo; ROSINGER, Chris; SANWALD, Erich; ARNOLD, Christian |
Die vorliegende Erfindung betrifft die Verwendung selektiv-insektizider und/oder akarizider Mittel, gekennzeichnet durch einen wirksamen Gehalt an einer Wirkstoffkombination umfassend (a) mindestens eine substituierte, cyclische Dicarbonylverbindung der Formel (I) in welcher W, X, Y und Z die in der Beschreibung angegebene Bedeutung haben und CDC für einen der in der Beschreibung genannten Dicarbonylreste steht, und (b) zumindest eine die Kulturpflanzen-Verträglichkeit verbessernde Verbindung aus der in der Beschreibung angegebenen Gruppe von Verbindungen zur Bekämpfung von Insekten und/oder Spinnentieren, sowie ein Verfahren zur Bekämpfung von Insekten und/oder Spinnentieren unter Einsatz der Mittel. |
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44 | Selective pyrazoline insecticides and fungicides | US633643 | 1990-12-21 | US5196546A | 1993-03-23 | John J. Delany |
Certain pyrazolines have been found to be useful as aphicides and fungicides. | ||||||
45 | S–二氟甲基高半胱胺酸,其製法及選擇性殺蟲劑 | TW078108035 | 1989-10-19 | TW150222B | 1991-01-21 | 石原照一; 津島忠彥 |
下式之化合物:□ (Ⅰ)其中R和R′各為氫或保護基,或其酸加成鹽,可作為選擇性殺蟲劑使用。 | ||||||
46 | ENANTIONSELECTIVE PROCESSES TO INSECTICIDAL 3-ARYL-3-TRIFLUOROMETHYL-SUBSTITUTED PYRROLIDINES | PCT/EP2012/069171 | 2012-09-28 | WO2013050301A1 | 2013-04-11 | SMEJKAL, Tomas; SMITS, Helmars; WENDEBORN, Sebastian, Volker; BERTHON, Guillaume; CASSAYRE, Jérôme, Yves; EL QACEMI, Myriem |
The present invention relates to processes for the enantio-selective preparation of spyrrolidine derivatives useful in the manufacture of pesticidally active compounds, as well as to intermedates in the processes. The processes include those comprising (a-i) reacting a compound of formula (Ia), formula (Ia), wherein P is alkyl, aryl or heteroaryl, each optionally substituted, wherein the heteroaryl is connected at P via a ring carbon atom; R1 is chlorodifluoromethyl or trifluoromethyl; R2 is aryl or heteroaryl, each optionally substituted; with a source of cyanide in the presence a chiral catalyst to give a compound of formula IIa, formula (IIa), wherein P, R1 and R2 are as defined for the compound of formula (Ia); and (a-ii) oxidising the compound of formula IIa with a peroxy acid, or peroxide in the presence of an acid to give a compound of formula (VI), formula (VI), wherein R1 and R2 are as defined for the compound of formula (Ia). |
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47 | INSECTICIDAL CARBAMATES EXHIBITING SPECIES-SELECTIVE INHIBITION OF ACETYLCHOLINESTERASE (ACHE) | PCT/US2008076108 | 2008-09-12 | WO2009036235A2 | 2009-03-19 | CARLIER PAUL R; BLOOMQUIST JEFFREY; PAULSON SALLY; WONG ERIC |
The present invention includes insecticidal carbamates that are useful, for example, for the control of insects, such as mosquitoes, which can be used in applications where exposure to and/or contact with humans is likely. The insecticides of the present invention include phenyl TV-methyl carbamates and compositions comprising them that exhibit species-selective inhibition of acetylcholinesterase (AChE) and are preferably toxic to mosquitoes but not humans. Of particular interest are compounds of Formula (I) and Formula (II): Compounds of Formula (I) and Formula (II) are especially suitable for insecticide treated nets and indoor residual spraying for mosquito control. | ||||||
48 | SELEKTIVE INSEKTIZIDE AUF BASIS VON HALOGENALKYLNICOTINSÄUREDERIVATEN, ANTHRANILSÄUREDIAMIDEN ODER PHTHALSÄUREDIAMIDEN UND SAFENERN | PCT/EP2005/007791 | 2005-07-18 | WO2006008108A2 | 2006-01-26 | FISCHER, Reiner; FISCHER, Rüdiger; FUNKE, Christian; HENSE, Achim; ANDERSCH, Wolfram; HUNGENBERG, Heike; THIELERT, Wolfgang; RECKMANN, Udo; WILLMS, Lothar; ARNOLD, Christian |
Die vorliegende Erfindung betrifft die Verwendung selektiv-insektizider Mittel, gekennzeichnet durch einen wirksamen Gehalt an einer Wirkstoffkombination umfassend: (a) (1) mindestens ein Halogenalkylnicotinsäurederivat der Formel (I), in welcher AA und R1A die in der Beschreibung angegebenen Bedeutungen haben, oder (2) mindestens ein Phthalsäurediamid der Formel (II), in welcher XB, R1B, R2B, R3B, L1B, L2B und L3B die in der Beschreibung angegebenen Bedeutungen haben, oder (3) mindestens ein Anthranilsäureamid der Formel (III), in welcher A1C, A2C, XC, R1C, R2C, R3C, R4C, R5C, R7C, R8C und R9C die in der Beschreibung angegebenen Bedeutungen haben, und (b) zumindest eine die Kulturpflanzen-Verträglichkeit verbessernde Verbindung aus der in der Beschreibung angegebenen Gruppe von Verbindungen, insbesondere Cloquintocet-mexyl, Isoxadifen-ethyl und Mefenpyr-diethyl zur Bekämpfung von Insekten und/oder Spinnentieren, sowie ein Verfahren zur Bekämpfung von Insekten und/oder Spinnentieren unter Einsatz der Mittel. |
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49 | ENHANCED BIOACTIVITY OF MAMMALIAN SOMATOTROPIN THROUGH SELECTIVE DEAMIDATION | PCT/US1986001860 | 1986-09-15 | WO1987001708A2 | 1987-03-26 | THE UPJOHN COMPANY |
Deamidated forms of mammalian somatotropins originally having an asparagine located between residues 96-101. These deamidated somatotropins have an increased bioactivity as compared to their native species. This invention particularly discloses a composition comprised of bovine somatotropin (bSt) compounds wherein the bSt has been modified by deamidation from the native state comprising a predominant electrophoretic species having an isoelectric point (pI) of 8.2 to a bioenhanced composition of bSt molecules having a predominant electrophoretic species with pI between 7.5 and 6.5. The preferred bovine somatotropin is that species in which the asparagine located between amino acid residues 96-101 has been modified to isoaspartic acid. Processes for the production of these bioenhanced compositions and for their use are also disclosed. | ||||||
50 | APPARATUS FOR SELECTIVELY DISPENSING FERTILIZER, PESTICIDE AND THE LIKE THROUGH A FLUID FLOW LINE | PCT/US2007/068852 | 2007-05-14 | WO2008024533A1 | 2008-02-28 | MESSINA, Steven |
An apparatus has a fluid flow portion that is introduced as part of a fluid flow continuum. The fluid flow portion is situated above a plurality of liquid-holding chambers. Each chamber forms a fluid flow continuum from the chamber through a tube-like structure that intersects the fluid flow portion. A control means is provided to set the fluid flow from the chamber at a determined level. An alternative embodiment provides an apparatus that is fully portable. |
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51 | SELECTIVE INSECTICIDES BASED ON HALOALKYLNICOTINIC ACID DERIVATIVES, ANTHRANILIC ACID DIAMIDES, OR PHTHALIC ACID DIAMIDES AND SAFENERS | PCT/EP2005007791 | 2005-07-18 | WO2006008108A3 | 2006-08-31 | FISCHER REINER; FISCHER RUEDIGER; FUNKE CHRISTIAN; HENSE ACHIM; ANDERSCH WOLFRAM; HUNGENBERG HEIKE; THIELERT WOLFGANG; RECKMANN UDO; WILLMS LOTHAR; ARNOLD CHRISTIAN |
The invention relates to the use of selective insecticides for controlling insects and/or arachnids. Said selective insecticides are characterized by an active moiety of an active substance combination comprising: (a) (1) at least one haloalkylnicotinic acid derivative of formula (I), wherein AA and R1A have the meanings indicated in the description, or (2) at least one phthalic acid diamine of formula (II), wherein XB, R1B, R2B, R3B, L1B, L2B, and L3B have the meanings indicated in the description, or (3) at least one anthranilic acid amide of formula (III), wherein A1C, A2C, XC, R1C, R2C, R3C, R4C, R5C, R7C, R8C, and R9C have the meanings indicated in the description, and (b) at least one compound that improves crop plant tolerance and is part of the group of compounds indicated in the description, especially cloquintocet-mexyl, isoxadifen-ethyl, and mefenpyr-diethyl. Also disclosed is a method for controlling insects and/or arachnids using the inventive insecticides. | ||||||
52 | ENHANCED BIOACTIVITY OF MAMMALIAN SOMATOTROPIN THROUGH SELECTIVE DEAMIDATION | PCT/US8601860 | 1986-09-15 | WO8701708A3 | 1987-08-13 | HARBOUR GARY C; HOOGERHEIDE JOHN G; GARLICK ROBERT L |
Deamidated forms of mammalian somatotropins originally having an asparagine located between residues 96-101. These deamidated somatotropins have an increased bioactivity as compared to their native species. This invention particularly discloses a composition comprised of bovine somatotropin (bSt) compounds wherein the bSt has been modified by deamidation from the native state comprising a predominant electrophoretic species having an isoelectric point (pI) of 8.2 to a bioenhanced composition of bSt molecules having a predominant electrophoretic species with pI between 7.5 and 6.5. The preferred bovine somatotropin is that species in which the asparagine located between amino acid residues 96-101 has been modified to isoaspartic acid. Processes for the production of these bioenhanced compositions and for their use are also disclosed. | ||||||
53 | SELEKTIVE INSEKTIZIDE AUF BASIS VON SUBSTITUIERTEN, CYCLISCHEN KETOENOLEN UND SAFENERN | EP05776440.9 | 2005-07-18 | EP1771067B1 | 2014-03-12 | FISCHER, Reiner; RECKMANN, Udo; ROSINGER, Christopher, Hugh; SANWALD, Erich; ARNOLD, Christian |
54 | Enhanced bioactivity of mammalian somatotropin through selective deamidation | EP86307767.3 | 1986-10-08 | EP0263206B1 | 1990-12-12 | Harbour, Gary C.; Hoogerheide, John G.; Garlick, Robert L. |
55 | SELEKTIVE INSEKTIZIDE AUF BASIS VON SUBSTITUIERTEN, CYCLISCHEN KETOENOLEN UND SAFENERN | EP05776440.9 | 2005-07-18 | EP1771067A1 | 2007-04-11 | FISCHER, Reiner; RECKMANN, Udo; ROSINGER, Christopher, Hugh; SANWALD, Erich; ARNOLD, Christian |
The invention relates to the use of selective insecticides for controlling insects and/or arachnids. Said insecticides are characterized by an active moiety of an active substance combination comprising (a) at least one compound of formula (I), wherein CKE, W, X, Y, and Z have the meaning indicated in the description, and (b) at least one compound which improves crop plant tolerance and is part of the group of compounds indicated in the description. Also disclosed is a method for controlling insects and/or arachnids using the inventive insecticides. | ||||||
56 | Selective Insecticides Based on Anthranilic Acid Diamides and Safeners | US12944074 | 2010-11-11 | US20110059991A1 | 2011-03-10 | Reiner Fischer; Rüdiger Fischer; Christian Funke; Achim Hense; Wolfram Andersch; Heike Hungenberg; Wolfgang Thielert; Udo Reckmann; Lothar Willms; Christian Arnold |
The present invention relates to the use of selective insecticidal compositions, characterized by an effective amount of an active compound combination comprising (a) (1) at least one haloalkylnicotinic acid derivative of the formula (I) in which AA and R1A are as defined in the description, or (2) at least one phthalic acid diamide of the formula (II) in which XB, R1B, R2B, R3B, L1B, L2B and L3B are as defined in the description, or (3) at least one anthranilamide of the formula (III) in which A1C, A2C, XC, R1C, R2C, R3C, R4C, R5C, R7C, R8C and R9C are as defined in the description, and (b) at least one crop plant compatibility-improving compound from the group of compounds given in the description, in particular cloquintocet-mexyl, isoxadifen-ethyl and mefenpyr-diethyl for controlling insects and/or arachnids, and a method for controlling insects and/or arachnids using the compositions. | ||||||
57 | Selective Insecticides Based on Anthranilic Acid Diamides and Safeners | US14095509 | 2013-12-03 | US20140087946A1 | 2014-03-27 | Reiner FISCHER; Rüdiger FISCHER; Christian FUNKE; Achim HENSE; Wolfram ANDERSCH; Heike HUNGENBERG; Wolfgang THIELERT; Udo RECKMANN; Lothar WILLMS; Christian ARNOLD |
The present invention relates to the use of selective insecticidal compositions, characterized by an effective amount of an active compound combination comprising (a) (1) at least one haloalkylnicotinic acid derivative of the formula (I) in which AA and R1A are as defined in the description, or (2) at least one phthalic acid diamide of the formula (II) in which XB, R1B, R2B, R3B, L1B, L2B and L3B are as defined in the description, or (3) at least one anthranilamide of the formula (III) in which A1C, A2C, XC, R1C, R2C, R3C, R4C, R5C, R7C, R8C and R9C are as defined in the description, and (b) at least one crop plant compatibility-improving compound from the group of compounds given in the description, in particular cloquintocet-mexyl, isoxadifen-ethyl and mefenpyr-diethyl for controlling insects and/or arachnids, and a method for controlling insects and/or arachnids using the compositions. | ||||||
58 | Selective insecticides based on substituted cyclic ketoenols and safeners | US11572400 | 2005-07-18 | US08202875B2 | 2012-06-19 | Reiner Fischer; Udo Reckmann; Christopher Hugh Rosinger; Erich Sanwald; Christian Arnold |
The present invention relates to the use of selective insecticidal compositions, characterized in that they comprise an effective amount of an active compound combination comprising (a) at least one compound of the formula (I) in which CKE, W, X, Y and Z are as defined in the description, and (b) at least one crop plant compatibility-improving compound, from the group of compounds mentioned in the description, for controlling insects and/or arachnids, and to a method for controlling insects and/or arachnids using the compositions. | ||||||
59 | Selective Insecticides Based on Substituted Cyclic Ketoenols and Safeners | US11572400 | 2005-07-18 | US20090012100A1 | 2009-01-08 | Reiner Fischer; Udo Reckmann; Christopher Hugh Rosinger; Erich Sanwald; Christian Arnold |
The present invention relates to the use of selective insecticidal compositions, characterized in that they comprise an effective amount of an active compound combination comprising (a) at least one compound of the formula (I) in which CKE, W, X, Y and Z are as defined in the description, and (b) at least one crop plant compatibility-improving compound, from the group of compounds mentioned in the description, for controlling insects and/or arachnids, and to a method for controlling insects and/or arachnids using the compositions. | ||||||
60 | Insecticidal n-(optionally substituted)-n'- substituted-n,n'-disubstituted hydrazine | JP9548787 | 1987-04-20 | JPS63267752A | 1988-11-04 | ADAMU CHIYAIITANGU SHIYU; DONARUDO UESUREI HAMUPU |