子分类：
| 序号 | 专利名 | 申请号 | 申请日 | 公开（公告）号 | 公开（公告）日 | 发明人 |
|---|---|---|---|---|---|---|
| 181 | Arylphenyl-substituted cyclic ketoenols | US11330601 | 2006-01-12 | US20060122061A1 | 2006-06-08 | Folker Lieb; Reiner Fischer; Alan Graff; Udo Schneider; Thomas Bretschneider; Christoph Erdelen; Wolfram Andersch; Mark-Wilhelm Drewes; Markus Dollinger; Ingo Wetcholowsky; Randy Myers |
| The present invention relates to novel arylphenyl-substituted cyclic ketoenols of the formula (I) in which X represents halogen, alkyl, alkoxy, alkenyloxy, alkylthio, alkylsulphinyl, alkylsulphonyl, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro, cyano or in each case optionally substituted phenyl, phenoxy, phenylthio, phenylalkoxy or phenylalkylthio, Y represents in each case optionally substituted cycloalkyl, aryl or hetaryl, Z represents hydrogen, halogen, alkyl, alkoxy, alkenyloxy, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro or cyano, CKE represents one of the groups in which A, B, D, G and Q1 to Q6 are each as defined in the description, to a plurality of processes for their preparation and to their use as pesticides and herbicides. | ||||||
| 182 | Herbicides | US10070767 | 2000-09-05 | US06894005B1 | 2005-05-17 | Thomas Maetzke; André Stoller; Sebastian Wendeborn; Henry Szczepanski |
| Compounds of formula wherein the substituents have the meanings given in claim 1, and agronomically tolerable salts, isomers and enantiomer of those compounds, are suitable for use as herbicides. | ||||||
| 183 | Arylphenyl-substituted cyclic ketoenols | US10730556 | 2003-12-08 | US06806264B2 | 2004-10-19 | Folker Lieb; Reiner Fischer; Alan Graff; Udo Schneider; Thomas Bretshneider; Christoph Erdelen; Wolfram Andersch; Mark Wilhelm Drewes; Markus Dollinger; Ingo Wetcholowsky; Randy Allen Myers |
| The present invention relates to novel arylphenyl-substituted cyclic ketoenols of the formula (I) in which X represents halogen, alkyl, alkoxy, alkenyloxy, alkylthio, alkylsulphinyl, alkylsulphonyl, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro, cyano or in each case optionally substituted phenyl, phenoxy, phenylthio, phenylalkoxy or phenylalkylthio, Y represents in each case optionally substituted cycloalkyl, aryl or hetaryl, W and Y independently of one another each represent hydrogen, halogen, alkyl, alkoxy, alkenyloxy, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro or cyano, CKE represents one of the groups in which A, B, D, G and Q1 to Q6 are each as defined in the description, to a plurality of processes for their preparation and to their use as pesticides and herbicides. | ||||||
| 184 | Spirocyclic dopamine receptor subtype ligands | US09242819 | 1999-02-24 | US06664258B1 | 2003-12-16 | Anton F. J. Fliri; Todd W. Butler |
| This invention relates to novel, pharmaceutically active compounds of formula (I) wherein a, b and R1 through R6 are as defined in the specification These compounds exhibit central dopaminergic activity and are useful in the treatment of CNS disorders. | ||||||
| 185 | Arylphenyl-substituted cyclic ketoenols | US10192361 | 2002-07-10 | US20030096806A1 | 2003-05-22 | Folker Lieb; Reiner Fischer; Alan Graff; Udo Schneider; Thomas Bretschneider; Christoph Erdelen; Wolfram Andersch; Mark Wilhelm Drewes; Markus Dollinger; Ingo Wetcholowsky; Dieter Feucht; Rolf Pontzen; Randy Allen Myers |
| The present invention relates to novel arylphenyl-substituted cyclic ketoenols of the formula (I) 1 in which X represents halogen, alkyl, alkoxy, alkenyloxy, alkylthio, alkylsulphinyl, alkylsulphonyl, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro, cyano or in each case optionally substituted phenyl, phenoxy, phenylthio, phenylalkoxy or phenylalkylthio, Y represents in each case optionally substituted cycloalkyl, aryl or hetaryl, W represents hydrogen, halogen, alkyl, alkoxy, alkenyloxy, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro or cyano, Z represents halogen, alkyl, alkoxy, alkenyloxy, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro or cyano, CKE represents one of the groups 2 in which A, B, D, G and Q1, S, Q6 are each as defined in the description, to a plurality of processes for their preparation and to their use as pesticides and herbicides. | ||||||
| 186 | Arylphenyl-substituted cyclic ketoenols | US10142325 | 2002-05-09 | US20030073851A1 | 2003-04-17 | Folker Lieb; Reiner Fischer; Alan Graff; Udo Schneider; Thomas Bretshneider; Christoph Erdelen; Wolfram Andersch; Mark Wilhelm Drewes; Markus Dollinger; Ingo Wetcholowsky; Randy Allen Myers |
| The present invention relates to novel arylphenyl-substituted cyclic ketoenols of the formula (I) 1 in which X represents halogen, alkyl, alkoxy, alkenyloxy, alkylthio, alkylsulphinyl, alkylsulphonyl, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro, cyano or in each case optionally substituted phenyl, phenoxy, phenylthio, phenylalkoxy or phenylalkylthio, Y represents in each case optionally substituted cycloalkyl, aryl or hetaryl, W and Y independently of one another each represent hydrogen, halogen, alkyl, alkoxy, alkenyloxy, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro or cyano, CKE represents one of the groups 2 nullin which A, B, D, G and Q1 to Q6 are each as defined in the description, to a plurality of processes for their preparation and to their use as pesticides and herbicides. | ||||||
| 187 | Arylphenyl-substituted cyclic ketoenols | US10137763 | 2002-05-02 | US20020188136A1 | 2002-12-12 | Folker Lieb; Reiner Fischer; Alan Graff; Udo Schneider; Thomas Bretschneider; Christoph Erdelen; Wolfram Andersch; Mark-Wilhelm Drewes; Markus Dollinger; Ingo Wetcholowsky; Randy Allen Myers |
| The present invention relates to novel arylphenyl-substituted cyclic ketoenols of the formula (I) 1 in which X represents halogen, alkyl, alkoxy, alkenyloxy, alkylthio, alkylsulphinyl, alkylsulphonyl, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro, cyano or in each case optionally substituted phenyl, phenoxy, phenylthio, phenylalkoxy or phenylalkylthio, Y represents in each case optionally substituted cycloalkyl, aryl or hetaryl, Z represents hydrogen, halogen, alkyl, alkoxy, alkenyloxy, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro or cyano, CKE represents one of the groups 2 nullin which A, B. D, G and Q1 to Q6 are each as defined in the description, to a plurality of processes for their preparation and to their use as pesticides and herbicides. | ||||||
| 188 | Aryl phenyl substituted cyclic ketoenols | US09646722 | 2001-01-02 | US06458965B1 | 2002-10-01 | Folker Lieb; Reiner Fischer; Alan Graff; Udo Schneider; Thomas Bretshneider; Christoph Erdelen; Wolfram Andersch; Mark Wilhelm Drewes; Markus Dollinger; Ingo Wetcholowsky; Randy Allen Myers |
| The present invention relates to novel arylphenyl-substituted cyclic ketonols of the formula (I) in which X represents halogen, alkyl, alkoxy, alkenyloxy, alkylthio, alkylsulphinyl, alkylsulphonyl, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro, cyano or in each case optionally substituted phenyl, phenoxy, phenylthio, phenylalkoxy or phenylalkylthio, Y represents in each case optionally substituted cycloalkyl, aryl or hetaryl, W and Y independently of one another each represent hydrogen, halogen, alkyl, alkoxy, alkenyloxy, halogenoalkyl, halogenoalkoxy, halogenoalkenyloxy, nitro or cyano, CKE represents one of the groups in which A, B, D, G and Q1 to Q6 are each as defined in the description, to a plurality of processes for their preparation and to their use as pesticides and herbicides. | ||||||
| 189 | 2- and 2,5-substituted phenylketoenols | US09809619 | 2001-03-15 | US20020010204A1 | 2002-01-24 | Folker Lieb; Reiner Fischer; Thomas Bretschneider; Michael Ruther; Alan Graff; Udo Schneider; Christoph Erdelen; Ulrike Wachendorff-Neuman; Wolfram Andersch; Andreas Turberg |
| The invention relates to novel phenyl-substituted cyclic ketoenols of the formula (I) 1 in which Het represents one of the groups 2 in which A, B, D, G, X and Z are each as defined in the description, to a plurality of processes and intermediates for their preparation, and to their use as pesticides. | ||||||
| 190 | Alkyl dihalogenated phenyl-substituted ketoenols useful as pesticides and herbicides | US08945664 | 1997-10-31 | US06316486B1 | 2001-11-13 | Folker Lieb; Hermann Hagemann; Arno Widdig; Michael Ruther; Reiner Fischer; Thomas Bretschneider; Christoph Erdelen; Ulrike Wachendorff-Neumann; Peter Dahmen; Markus Dollinger; Hans-Joachim Santel; Alan Graff; Wolfram Andersch; Norbert Mencke; Andreas Turberg |
| The present invention relates to new compounds of the formula (I) in which X represents halogen, Y represents halogen or alkyl and Z represents halogen or alkyl, with the proviso that always one of the radicals Y and Z represents halogen while the other represents alkyl, and Het represents one of the groups in which A, B, D and G have the meanings given in the description, to a plurality of processes for their preparation and to their use as pesticides and herbicides. | ||||||
| 191 | 2-and 2,5-substituted phenylketoenols | US09548129 | 2000-04-12 | US06255342B1 | 2001-07-03 | Folker Lieb; Reiner Fischer; Thomas Bretschneider; Michael Ruther; Alan Graff; Udo Schneider; Christoph Erdelen; Ulrike Wachendorff-Neumann; Wolfram Andersch; Andreas Turberg |
| The invention relates to novel phenyl-substituted cyclic ketoenols of the formula (I) in which Het represents one of the groups in which A, B, D, G, X and Z are each as defined in the description, to a plurality of processes and intermediates for their preparation, and to their use as pesticides. | ||||||
| 192 | Substituted phenyl keto enols as pesticides and herbicides | US09550105 | 2000-04-14 | US20010004629A1 | 2001-06-21 | Volker Lieb; Hermann Hagemann; Arno Widdig; Michael Ruther; Reiner Fischer; Thomas Bretschneider; Christoph Erdelen; Ulrike Wachendorff-Neumann; Alan Graff; Udo Schneider |
| The present invention relates to novel compounds of the formula (I) 1 in which Het represents one of the groups 2 in which A, B, D, G, V, W, X, Y and Z are as defined in the description, processes and intermediates for their preparation, and to their use as pesticides and herbicides. | ||||||
| 193 | 2-and 2,5-substituted phenylketoenols | US230653 | 1999-01-28 | US06114374A | 2000-09-05 | Folker Lieb; Reiner Fischer; Thomas Bretschneider; Michael Ruther; Alan Graff; Udo Schneider; Christoph Erdelen; Ulrike Wachendorff-Neumann; Wolfram Andersch; Andreas Turberg |
| The invention relates to novel phenyl-substituted cyclic ketoenols of the formula (I) ##STR1## in which Het represents one of the groups ##STR2## in which A, B, D, G, X and Z are each as defined in the description, to a plurality of processes and intermediates for their preparation, and to their use as pesticides. | ||||||
| 194 | 3-aryl-4-hydroxy-.DELTA..sup.3 -dihydrothiophenone derivatives | US716361 | 1996-09-18 | US5945444A | 1999-08-31 | Reiner Fischer; Jacques Dumas; Thomas Bretschneider; Christoph Erdelen; Ulrike Wachendorff-Neumann |
| The present invention relates to novel 3-aryl-4-hydroxy-.DELTA..sup.3 -dihydrothiophenone derivatives of the formula (I) ##STR1## in which A, B, G, S, X, Y, Z and n have the meaning given in the description, to processes for their preparation, to novel intermediates and to the use of the compounds of the formula (I) as agents for controlling pests. | ||||||
| 195 | Asymmetric synthesis and catalysis with chiral heterocyclic compounds | US6178 | 1998-01-13 | US5936127A | 1999-08-10 | Xumu Zhang |
| This invention relates to chiral heterocyclic compounds useful for asymmetric synthesis and catalysis. More particularly, the invention relates to chiral heterocyclic phosphine, sulfur, and nitrogen compounds for asymmetric synthesis and catalysis in the production of enantiomerically pure products. | ||||||
| 196 | Process for preparing .gamma.-mercaptocarboxylic acid derivatives | US297756 | 1994-08-30 | US5534651A | 1996-07-09 | Wilhelm Quittmann; John McGarrity |
| .gamma.-Mercaptocarboxylic acids and their derivatives, in particular esters and amides, are prepared from .gamma.-butyrolactones via the corresponding thiolactones. The thiolactones are obtained by reaction of a .gamma.-lactone with thiocarboxylates in polar solvents and are converted by ring opening using nucleophilic reagents, such as, alkali metal alkoxides, into the .gamma.-mercaptocarboxylic acid derivatives. These are intermediates, for example, for the synthesis of leucotriene antagonists. | ||||||
| 197 | Hindered linking agents and methods | US796048 | 1991-11-20 | US5183904A | 1993-02-02 | Stephen F. Carroll; Dane A. Goff |
| Novel compounds and methods for the formation of disulfide linkages are presented. The novel compounds employed are substituted 2-iminothiolane hydrohalide linking agents of the following formula (I): ##STR1## wherein, X is halogen;R.sub.1 is COOR.sub.5 ; halogen; nitro; unsubstituted or halogenated C.sub.1-8 alkyl; unsubstituted or halogenated C.sub.1-8 alkoxy; unsubstituted or halogenated C.sub.2-8 alkenyl; unsubstituted or halogenated C.sub.2-8 alkynyl; unsubstituted C.sub.3-8 cycloalkyl; unsubstituted aryl; aryl substituted with 1 to 3 substituents selected from halogen, amino, unsubstituted or halogenated C.sub.1-8 alkyl, or unsubstituted or halogenated C.sub.1-8 alkoxy; unsubstituted heterocycle; or heterocycle substituted with 1 to 3 substituents selected from amino, halogen, unsubstituted or halogenated C.sub.1-8 alkyl, or unsubstituted or halogenated C.sub.1-8 alkoxy;each of R.sub.2, R.sub.3 and R.sub.4 is independently hydrogen or selected from the values of R.sub.1 ; orR.sub.1 and R.sub.2 together form a C.sub.2-5 alkylene bridge, unsubstituted or substituted with one to five C.sub.1-4 alkyl groups; orR.sub.1 or R.sub.2 together with R.sub.3 form a C.sub.1-5 alkylene bridge, unsubstituted or substituted with one to five C.sub.1-4 alkyl groups; andR.sub.5 is hydrogen or C.sub.1-8 alkyl.Also included in the invention are methods for covalently linking two species, which methods comprise reacting one or both of the two species with a crosslinking agent of the above formula (I) and mixing the two species together. The resulting conjugated species containing the linking group are also included in the invention.Further included in the invention is the use of a quenching agent which allows direct measurement of the reaction of 2-iminothiolanes with nucleophilic groups. | ||||||
| 198 | Certain substituted naphthofurans with anti-tumor properties | US401612 | 1989-08-28 | US5008286A | 1991-04-16 | Kenneth W. Bair |
| The present invention relates to compounds of formula (I)ArCH.sub.2 R.sup.1 (I)or a monomethyl or monethyl ether thereof (the compound of formula (I) including these ethers may contain no more than 29 carbon atoms in total); ethers, esters thereof; acide addition salts thereof; wherein Ar is a fused tricyclic aromatic ring system containing a maximum of 14 ring atoms and at least one heteroatom or a fused pentacyclic ring system with at least 4 aromatic rings containing a maximum of 22 ring atoms and at least one heteroatom; or a substituted derivative thereof; for either the tricyclic or pentacyclic ring system there is a maximum of one heteroatom for each ring present but preferably only one or two of the rings contain a heteroatom; the rings forming the tricyclic or the pentacyclic ring system contain five or six atoms; the heteroatoms are conveniently nitrogen, phosphorus, oxygen, sulfur or selenium; suitably the heteroatom is oxygen, sulfur or nitrogen; the tricyclic or the pentacyclic ring system should be planar or deviate only slightly from planarity; suitably the ring system is aromatic or contains one non-aromatic ring; preferably the ring system is aromatic; nitrogen atoms contained in five-membered rings are substituted by hydrogen, methyl or ethyl; R.sup.1 contains not more than eight carbon atoms and is a group ##STR1## wherein m is 0 or 1; R.sup.5 is hydrogen;R.sup.6 and R.sup.7 are the same or different and each is hydrogen or C.sub.1-5 alkyl optionally substituted by hydroxy;R.sup.8 and R.sup.9 are the same or different and each is hydrogen or C.sub.1-3 alkyl; ##STR2## is a five or six-membered saturated carbocyclic ring; R.sup.10 is hydrogen, methyl or hydroxymethyl;R.sup.11, R.sup.12 and R.sup.13 are the same or different and each is hydrogen or methyl;R.sup.14 is hydrogen, methyl, hydroxy, or hydroxymethyl.The compounds have biocidal properties. | ||||||
| 199 | Aryl-substituted thiophene 3-ols, derivatives and analogs useful as lipoxgenase inhibitors | US397325 | 1989-08-22 | US4999436A | 1991-03-12 | Bruce E. Witzel; Debra L. Allison; Charles G. Caldwell; Kathleen Rupprecht |
| Aryl substituted thiophenes 3-ols, its dihydro derivatives, 1-oxide and 1,1-dioxide analogs, as well as aryl substituted furans, are 5-lipoxygenase inhibitors useful in the treatment of inflammation and other leukotriene-mediated diseases. | ||||||
| 200 | Dibenzothiphene and naphthalenethiophene derivatives | US399713 | 1989-08-25 | US4965285A | 1990-10-23 | Kenneth W. Bair |
| The present invention relates to compounds of formula (I)ArCH.sub.2 R.sup.1 (I)or a monomethyl or monoethyl ether thereof (the compound of formula (I) including these ethers may contain no more than 29 carbon atoms in total); ethers, esters thereof; acid addition salts thereof; wherein Ar is a fused tricyclic aromatic ring system containing a maximum of 14 ring atoms and at least one heteroatom or a fused pentacyclic ring system with at least 4 aromatic rings containing a maximum of 22 ring atoms and at least one heteroatom; or a substituted derivative thereof; for either the tricyclic or pentacyclic ring system there is a maximum of one heteroatom for each ring present but preferably only one or two of the rings contain a heteroatom; the rings forming the tricyclic or the pentacyclic ring system contain five or six atoms; the heteroatoms are conveniently nitrogen, phosphorus, oxygen, sulfur or selenium; suitably the heteroatom is oxygen, sulfur or nitrogen; the tricyclic or the pentacyclic ring system should be planar or deviate only slightly from planarity; suitably the ring system is aromatic or contains one non-aromatic ring; preferably the ring system is aromatic; nitrogen atoms contained in five-membered rings are substituted by hydrogen, methyl or ethyl; R.sup.1 contains not more than eight carbon atoms and is a group ##STR1## wherein m is 0 or 1; R.sup.5 is hydrogen;R.sup.6 and R.sup.7 are the same or different and each is hydrogen or C.sub.1-5 alkyl optionally substituted by hydroxy;R.sup.8 and R.sup.9 are the same or different and each is hydrogen or C.sub.1-3 alkyl; ##STR2## is a five or six-membered saturated carbocyclic ring; R.sup.10 is hydrogen, methyl or hydroxymethyl;R.sup.11, R.sup.12 and R.sup.13 are the same or different and each is hydrogen or methyl;R.sup.14 is hydrogen, methyl, hydroxy, or hydroxymethyl. | ||||||
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