| 序号 | 专利名 | 申请号 | 申请日 | 公开（公告）号 | 公开（公告）日 | 发明人 |
|---|---|---|---|---|---|---|
| 101 | 22 harogenmechiru 1*44 benzoshijiazepinnoseiho | JP12235975 | 1975-10-09 | JPS5165786A | 1976-06-07 | HORUSUTO TSUOIGUNERU; BORUFUGANGU MIRUKOFUSUKII; HANSU RIIPUMAN; JIIKUFURIITO FUNKE; BERUNERU SHUTOYUUMERU; RORUFU HYUTSUSHENSU |
| 102 | METHOD FOR PREPARATION OF CERTAIN THIOACETAMIDES | EP15174514.8 | 2015-06-30 | EP3112344A1 | 2017-01-04 | ZARAGOZA DOERWALD, Florencio |
The invention discloses a method for the preparation of certain thioacetamides with sulfur chlorides starting from certain methylketones, and their use in the preparation of certain 1,5 disubstituted tetrazoles, which allows the preparation of said tetrazoles from readily available compounds such as acetophenone and similar compounds. |
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| 103 | Method of Preparing a Halogenated Compound | EP03003782.4 | 1998-12-10 | EP1319642B1 | 2008-03-26 | Suzuki, Daisuke; Kikuchi, Ryo; Yasui, Masaru |
| 104 | Process to prepare aryltriazolinones and novel intermediates thereto | EP04005348.0 | 2000-10-12 | EP1440968A1 | 2004-07-28 | Goudar, Jaidev S |
A process is described for preparing 1-aryltriazolinones of formula (I) useful in the production of commercial herbicides, by: condensing a hydrazonoyl derivative of formula (A) with one or more ring-forming agent in formula (A), where W is halogen, -NCO, -OSO2CH3, -OSO2CF3, or -OSO2(p-CH3Ph); and X, Y, Z, and R1 are fully described herein. Certain compounds of formula (A) are novel compositions of matter. The process as described herein has utility in providing compounds of formula (I) in unexpectedly high yield and purity.
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| 105 | Method of Preparing a Halogenated Compound | EP03003782.4 | 1998-12-10 | EP1319642A3 | 2003-12-03 | Suzuki, Daisuke; Kikuchi, Ryo; Yasui, Masaru |
A halogenated compound of formula A-X is prepared by reacting in an organic solvent at least one halogenatihg agent selected from halogenating agents of formula |
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| 106 | Method of Preparing a Halogenated Compound | EP03003782.4 | 1998-12-10 | EP1319642A2 | 2003-06-18 | Suzuki, Daisuke; Kikuchi, Ryo; Yasui, Masaru |
A halogenated compound of formula A-X is prepared by reacting in an organic solvent at least one halogenatihg agent selected from halogenating agents of formula
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| 107 | N-ACYL-N-PHENYLTETRAHYDROPHTHALAMIC ACID DERIVATIVE, PRODUCTION THEREOF, AND HERBICIDE CONTAINING THE SAME AS ACTIVE INGREDIENT | EP91914759.5 | 1991-08-21 | EP0496900A1 | 1992-08-05 | TAKEMATU, Tetuo, 612, Mine-machi; KUME, Takashi, 11-4, Fujimi-machi; KOMATA, Takeo, 11-19, Higashida-cho; SUZUKI, Kiyoshi, 775-23, Hiramatu-honcho; MINEZAKI, Matsue; SIRAKAWA, Yumiko, 19-12, Arai-cho; MORI, Kaoru |
An N-acyl-N-phenyltetrahydrophthalamic acid derivative represented by general formula (I), a process for producing the same, and a herbicide containing the same as the active ingredient: wherein X and Y represent each independently hydrogen or halogen; R¹ represents hydrogen, halogen, lower alkoxy, lower alkenyloxy, lower alkynyloxy, lower alkoxyalkoxy or lower alkoxycarbonylalkoxy; R² represents lower alkyl, halogenated lower alkyl, or (un)substituted phenyl; and R³ represents lower alkoxy, lower alkenyloxy, lower alkynyloxy, lower alkoxyalkoxy, benzyloxy, or lower alkoxycarbonylalkoxy. The herbicide is widely applicable to upland fields, paddy fields, orchards, pastures, turfs, forests, non-crop lands and so forth, and is highly safe to crops, thus proving very useful.
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| 108 | IMINE COMPOUND AND USE THEREOF | PCT/CN2022118920 | 2022-09-15 | WO2023051261A1 | 2023-04-06 | WU HONGFEI; XU JINGBO; SUN JUN; HAN JINLONG; LIU SHAOWU; XIE XISHAN; GUO CHUNXIAO; XU LIBAO; CHENG XUEMING; YU HAIBO |
| The present invention belongs to the field of insecticides and acaricides, and specifically relates to an imine compound and the use thereof. The structure is as represented by general formula I, wherein each substituent in the formula is defined in the description. The compound of general formula I has excellent insecticidal and acaricidal activities, and can be used for preventing and controlling various pest insects or pest mites. | ||||||
| 109 | METHOD OF MAKING COVALENT CONJUGATES WITH HIS-TAGGED PROTEINS | PCT/EP2008/056361 | 2008-05-23 | WO2008145609A1 | 2008-12-04 | AUER, Manfred; HINTERSTEINER, Martin; KIMMERLIN, Thierry |
The present invention refers to novel agents for covalently conjugating His-tagged proteins, to covalent conjugates of His-tagged proteins and to methods of making such conjugates. |
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| 110 | CATALYSTS CONTAINING N-PYRROLYL SUBSTITUTED NITROGEN DONORS | PCT/US0113643 | 2001-04-27 | WO0183571A3 | 2002-05-23 | MOODY LESLIE SHANE; MACKENZIE PETER BORDEN; KILLIAN CHRISTOPHER MOORE; LAVOIE GINO GEORGES; PONASIK JAMES ALLEN JR; SMITH THOMAS WILLIAM; PEARSON JASON CLAY; BARRETT ANTHONY GERARD MARTIN; COATES GEOFFREY WILLIAM |
| Catalyst compositions useful for the polymerization or oligomerization of olefins are disclosed. Certain of the catalyst compositions comprise N-pyrrolyl substituted nitrogen donors. Also disclosed are processes for the polymerization or oligomerization of olefins using the catalyst compositions. | ||||||
| 111 | CATALYSTS CONTAINING N-PYRROLYL SUBSTITUTED NITROGEN DONORS | PCT/US2001/013643 | 2001-04-27 | WO01083571A2 | 2001-11-08 | |
| Catalyst compositions useful for the polymerization or oligomerization of olefins are disclosed. Certain of the catalyst compositions comprise N-pyrrolyl substituted nitrogen donors. Also disclosed are processes for the polymerization or oligomerization of olefins using the catalyst compositions. | ||||||
| 112 | PROCESS TO PREPARE ARYLTRIAZOLINONES AND NOVEL INTERMEDIATES THERETO | PCT/US0028240 | 2000-10-12 | WO0127092A3 | 2001-10-25 | GOUDAR JAIDEV S |
| A process is described for preparing 1-aryltriazolinones of formula (I) useful in the production of commercial herbicides, by: i) carbonylating an amidrazone of formula (A) with one or more carbonylating agent, or ii) condensing a hydrazonoyl derivative of formula (A) with one or more ring-forming agent in formula (A), where W, X, Y, Z, and R<1> are fully described herein. Preferred are those where W is halogen or -NHR where R is hydrogen or haloalkyl; X and Y are independently selected from hydrogen, chloro, or fluoro; Z is hydrogen, bromo, iodo, nitro, amino, or methylsulfonylamino; and R<1> is methyl. Certain compounds of formula (A) are novel compositions of matter. The process as described herein has utility in providing compounds of formula (I) in unexpectedly high yield and purity. | ||||||
| 113 | PYRIMIDIN-4-ENAMINE AS FUNGICIDE | PCT/EP9908447 | 1999-11-04 | WO0031082A8 | 2000-08-03 | WALTER HARALD |
| Novel pyrimidine derivatives of formula (I), as well as possible isomers and mixtures of isomers thereof. The novel compounds have plant-protective properties and are suitable for protecting plants against infestations by phytopathogenic microorganisms and insecticidal attack. | ||||||
| 114 | PYRIMIDIN-4-ENAMINE AS FUNGICIDE | PCT/EP1999/008447 | 1999-11-04 | WO00031082A1 | 2000-06-02 | |
| Novel pyrimidine derivatives of formula (I), as well as possible isomers and mixtures of isomers thereof, wherein A is a 5- or 6-membered ring which may be saturated or unsaturated, aromatic or non-aromatic and which may contain no hetero atoms or 1-3 hetero atoms O, S and/or N, each in the free form or in salt form; R1, R2 and R3 are each independently of the other hydrogen; halogen; C1-C8alkyl, C2-C8alkenyl or C2-C8alkinyl which are unsubstituted or mono- to tri-substituted by C3-C6cycloalkyl, halogen, C1-C6alkoxy, C1-C6alkylthio or C1-C6haloalkoxy; O-C1-C6alkyl, O-C2-C6alkenyl, O-C2-C6alkynyl, S-C1-C6alkyl, S-C2-C6alkenyl or S-C2-C6alkynyl, which are unsubstituted or mono- to tri-substituted by C3-C6cycloalkyl, halogen, C1-C6alkoxy or C1-C6haloalkoxy; cyano; nitro; or trimethylsilyl; provided that R1, R2 and R3 are not hydrogen at the same time; R4 is C1-C8alkyl, C2-C8alkenyl or C2-C8alkinyl which are unsubstituted or mono- to tri-substituted by C3-C6cycloalkyl, halogen, cyano, nitro, CO-C1-C4alkyl, COO-C1-C4alkyl, CO-aryl, COO-aryl, C1-C6alkoxy or C1-C6haloalkoxy; C3-C6cycloalkyl which is unsubstituted or mono- to tri-substituted by C1-C6alky, C1-C6haloalkyl, halogen, cyano, C1-C6alkoxy or C1-C6haloalkoxy; phenyl or benzyl, in which the phenyl group is unsubstituted or mono- to pentasubstituted by halogen, cyano, nitro, C1-C8alkyl, C2-C8alkenyl, C2-C8alkinyl, C1-C6alkoxy, C1-C6haloalkoxy or C1-C6haloalkyl; NHR7; SR7 or OR7; R<5> is C1-C8alky, C2-C8alkenyl or C2-C8alkinyl which are unsubstituted or mono- to tri-substituted by C3-C6cycloalkyl, halogen, cyano, nitro, CO-C1-C4alkyl, COO-C1-C4alkyl, CO-aryl, COO-aryl, C1-C6alkoxy, C1-C6alkylthio or C1-C6haloalkoxy; C3-C6cycloalkyl which is unsubstituted or mono- to tri-substituted by C1-C6alkyl, halogen, cyano, C1-C6alkoxy, C1-C6haloalkyl or C1-C6haloalkoxy; R6 is hydrogen; C1-C8alkyl, C2-C8alkenyl or C2-C8alkinyl which are unsubstituted or mono- to tri-substituted by C3-C6cycloalkyl, halogen, cyano, nitro, CO-C1-C4alkyl, COO-C1-C4alkyl, CO-aryl, COO-aryl, C1-C6alkoxy, C1-C6alkylthio or C1-C6haloalkoxy; C3-C6cycloalkyl which is unsubstituted or mono- to tri-substituted by C1-C6alkyl, halogen, cyano, C1-C6alkoxy, C1-C6haloalkyl or C1-C6haloalkoxy; O-C1-C6alkyl, O-C2-C6alkenyl, O-C2-C6alkynyl, S-C1-C6alkyl, S-C2-C6alkenyl or S-C2-C6alkynyl which are unsubstituted or mono- to tri-substituted by C3-C6cycloalkyl, cyano, halogen, C1-C6alkoxy or C1-C6haloalkoxy; aryl or heteroaryl which are unsubstituted or mono- to tri-substituted by halogen, cyano, nitro, C1-C6alkyl, C1-C6haloalkyl, C1-C6alkoxy or C1-C6haloalkoxy; CO-C1-C6alkyl; CO-C1-C6alkyl-O-C1-C6alkyl; CO-C1-C6haloalkyl; CO-heteroaryl; SO2-C1-C6alkyl; SO2-ary | ||||||
| 115 | PROCESS FOR PRODUCTION OF 1-ARYL-5-(TRIFLUOROMETHYL)-1H- TETRAZOLES | EP04788473.9 | 2004-09-30 | EP1671945A1 | 2006-06-21 | HAGIYA, K., Toyo Kasei Kogyo Company Limited; SATO, Yasuhiro, Toyo Kasei Kogyo Company Limited; KOGURO, Kiyoto, Toyo Kasei Kogyo Company Limited; MITSUI, Sunao, Toyo Kasei Kogyo Company Limited |
The present invention relates to a process for producing an N-aryl-2,2,2-trifluoroacetimidoyl chloride represented by Formula (2):
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| 116 | Process for the preparation of 2-aryl-5-(perfluoroalkyl)pyrrole compounds from N-[1-chloro-1-(perfluoroalkyl)methyl]arylimidoyl chloride compounds | EP00301810.8 | 2000-03-06 | EP1035113A3 | 2001-08-08 | Kameswaran, Venkataraman |
There is provided a process for the preparation of 2-aryl-5-(perfluoroalkyl)pyrrole compounds of formula I from N-[1-chloro-1-(perfluoroalkyl)methyl]arylimidoyl chloride compounds. The 2-aryl-5-(perfluoroalkyl)pyrrole compounds are useful for the control of insect and acarid pests, and may also be used to prepare other pesticidal arylpyrrole compounds. In addition, the present invention provides compounds which are useful as intermediates in the preparation of arylpyrrole compounds. |
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| 117 | Process for the preparation of 2-aryl-5-(perfluoroalkyl)pyrrole compounds from N-[1-chloro-1-(perfluoroalkyl)methyl]arylimidoyl chloride compounds | EP00301810.8 | 2000-03-06 | EP1035113A2 | 2000-09-13 | Kameswaran, Venkataraman |
There is provided a process for the preparation of 2-aryl-5-(perfluoroalkyl)pyrrole compounds of formula I from N-[1-chloro-1-(perfluoroalkyl)methyl]arylimidoyl chloride compounds. The 2-aryl-5-(perfluoroalkyl)pyrrole compounds are useful for the control of insect and acarid pests, and may also be used to prepare other pesticidal arylpyrrole compounds. In addition, the present invention provides compounds which are useful as intermediates in the preparation of arylpyrrole compounds.
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| 118 | N-ACYL-N-PHENYLTETRAHYDROPHTHALAMIC ACID DERIVATIVE, PRODUCTION THEREOF, AND HERBICIDE CONTAINING THE SAME AS ACTIVE INGREDIENT | EP91914759.5 | 1991-08-21 | EP0496900B1 | 1996-05-29 | TAKEMATU, Tetuo, 612, Mine-machi; KUME, Takashi, 11-4, Fujimi-machi; KOMATA, Takeo, 11-19, Higashida-cho; SUZUKI, Kiyoshi, 775-23, Hiramatu-honcho; MINEZAKI, Matsue; SIRAKAWA, Yumiko, 19-12, Arai-cho; MORI, Kaoru |
| An N-acyl-N-phenyltetrahydrophthalamic acid derivative represented by general formula (I), a process for producing the same, and a herbicide containing the same as the active ingredient: wherein X and Y represent each independently hydrogen or halogen; R1 represents hydrogen, halogen, lower alkoxy, lower alkenyloxy, lower alkynyloxy, lower alkoxyalkoxy or lower alkoxycarbonylalkoxy; R2 represents lower alkyl, halogenated lower alkyl, or (un)substituted phenyl; and R3 represents lower alkoxy, lower alkenyloxy, lower alkynyloxy, lower alkoxyalkoxy, benzyloxy, or lower alkoxycarbonylalkoxy. The herbicide is widely applicable to upland fields, paddy fields, orchards, pastures, turfs, forests, non-crop lands and so forth, and is highly safe to crops, thus proving very useful. | ||||||
| 119 | N-ACYL-N-PHENYLTETRAHYDROPHTHALAMIC ACID DERIVATIVE, PRODUCTION THEREOF, AND HERBICIDE CONTAINING THE SAME AS ACTIVE INGREDIENT | EP91914759.5 | 1991-08-21 | EP0496900A4 | 1994-01-05 | TAKEMATU, Tetuo, 612, Mine-machi; KUME, Takashi, 11-4, Fujimi-machi; KOMATA, Takeo, 11-19, Higashida-cho; SUZUKI, Kiyoshi, 775-23, Hiramatu-honcho; MINEZAKI, Matsue; SIRAKAWA, Yumiko, 19-12, Arai-cho; MORI, Kaoru |
| 120 | Herbicidal 4,5-dihydro-1H-1,2,4-triazole-3-carboxamide derivatives | EP87303656.0 | 1987-04-24 | EP0290682B1 | 1992-07-01 | Shida, Takafumi; Kubota, Yoshikazu; Ichinose, Isao; Yamazaki, Shiro; Shinkawa, Hiroyasu |
