| 序号 | 专利名 | 申请号 | 申请日 | 公开（公告）号 | 公开（公告）日 | 发明人 |
|---|---|---|---|---|---|---|
| 21 | CNS 흥분제 | KR1019810003719 | 1981-10-02 | KR1019830007594A | 1983-11-04 | 라인하르트피터스타인 |
| 내용없음 | ||||||
| 22 | CNS 흥분제 및 항 고혈압제 | KR1019810003720 | 1981-10-02 | KR1019830007595A | 1983-11-04 | 레인하르드트페터스타인 |
| 내용없음 | ||||||
| 23 | Emitting device and device used therein | JP2003546416 | 2002-11-15 | JP2005510036A | 2005-04-14 | ピロウ，ジョナサン，ニジェール，ジェラルド; フランプトン，マイケル，ジョン |
| 下記の化合物（Ｉ）、（ＩＩ）又は（ＩＩＩ）の少なくとも１つを含有する発光装置。
【化１】 【化２】 【化３】 ここで、Ｒ 1及びＲ 2は、同じか異なり、Ｈを含まない有機置換基である。 ここで、Ｒ 3及びＲ 5は、ハロゲン及びＨを含まない有機置換基から選択される。 ここで、Ｒ 4 、Ｒ 6 、Ｒ 7 、Ｒ 8 、Ｒ 9及びＲ 10は、Ｈ、ハロゲン及び有機置換基からそれぞれ独立して選択される。 ここで、Ｒ 1 、Ｒ 2 、Ｒ 3 、Ｒ 4 、Ｒ 5 ，Ｒ 6 、Ｒ 7 、Ｒ 8 、Ｒ 9 、及びＲ 10が還系を形成するために選択的に縮合される。 ただし、Ｒ 3及びＲ 5の１つが縮合環の一部ではなく、また、Ｒ 1及びＲ 2が環を形成するために縮合しない。 ここで、Ｒ 3及びＲ 4の、又はＲ 5及びＲ 6両方ではなくどちらかは、環を形成するために互いに縮合される。 |
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| 24 | Di - or triaza - spiro [4,5] decane derivative | JP16194399 | 1999-06-09 | JP3369123B2 | 2003-01-20 | アンドレア・セスラ; ゲオ・アダム; ザビーネ・コルツェヴスキ; シュテファン・レーヴァー; フランソワ・ジェンク; ユルゲン・ヴィッヒマン |
| 25 | The novel heterocyclic compounds, their use in the treatment of these manufacturing methods and pharmaceutical compositions containing them, as well as diabetes and related diseases | JP53930797 | 1997-06-30 | JP2002515874A | 2002-05-28 | ガーラム、ランガ・マッドハバン; チャクラバルティ、ラニャン; パカラ、サルマ・ケー・エス; パラセリ、ラオ・ベーマ; ラマニャム、ラジャゴパラン; ローライ、ビッダヤ・ブースハン; ローライ、ブライ・ブースハン |
| (57)【要約】 | ||||||
| 26 | Di- or triaza-spiro[4,5]decane derivative | JP16194399 | 1999-06-09 | JP2000026466A | 2000-01-25 | ADAM GEO; CESURA ANDREA; JENCK FRANCOIS; KOLCZEWSKI SABINE; ROEVER STEPHAN; WICHMANN JUERGEN |
| PROBLEM TO BE SOLVED: To obtain a novel compound that is an agonist and antagonist of Orphanin FQ(OFQ) receptor and is useful for treatment of psychological disorder, neurological disorder and physiological disorder. SOLUTION: This is a new compound represented by formula I [R1 is a (substituted) 6-10C cycloalkyl, decahydro-naphthalen-1-yl, indan-1-yl, or the like; R2 is H, a lower alkyl, =O, or a (substituted) phenyl; group A is a (substituted) cyclohexyl or phenyl; X is -CH(OH)-, -C(O)- or the like; Y is -CH2-, -CH=, -N= or the like; a and b mean actual additive bonds], typically (RS)-8-(cis-4- isopropyl-cyclohexyl)-1-phenyl-1,8-diaza-spiro[4.5]decan-4-ol. The compound of formula I is prepared by reductive amination of a compound of formula II with a compound of formula II. | ||||||
| 27 | Chloroacetamide derivatives | JP1953583 | 1983-02-08 | JPH0645617B2 | 1994-06-15 | カ−ル・ゼツキンガ−; カ−ルハインツ・ミルツナ−; フレツド・ク−ネン |
| 28 | JPH0564634B2 - | JP5361485 | 1985-03-18 | JPH0564634B2 | 1993-09-16 | SHIMIZU NOBORU; ISHIWATARI HIROYUKI; KUNIEDA HISASHI; OOTA TOMIO; ISHIHAMA HIROSHI; UCHIDA YASUYOSHI |
| 29 | JPH0149353B2 - | JP18640985 | 1985-08-23 | JPH0149353B2 | 1989-10-24 | OKAZAKI MITSUO; YAMAGUCHI TERUHIRO; SASAKI MASAOMI |
| 30 | Heterocyclic thioalanine derivative | JP8387786 | 1986-04-11 | JPS62240663A | 1987-10-21 | MORITA YOSHIMI; HOSHIIDE YASUO; TANIGUCHI SEIRO; OKADA KAZUO; ANDO RYOICHI; TAKASHIMA JUNKO |
| NEW MATERIAL:A compound of formula I (P is formula VI-VIII; Q is O, S, NR<2>; Z is N, CR<8>; R<1>-R<8> are H, alkyl, further R<1> is H, alkyl; R<3> and R<4> incorporate to form alicyclic or aromatic ring; dotted line represents a bond existing in some cases; A is H, amino acid or oligopeptide which may have protecting group of the residue after removing OH from terminal CO2H or protecting group, B is OH, amino acid or oligopeptide residue which may have protecting groups after removing H from terminal NH2, protecting group). EXAMPLE:S-(2-Methyl-1,3,4-thiadiazol-5-yl)-D-cysteine. USE:A synthetic intermediate of inhibitor of cell wall biosynthesis and antibacterial agent. PREPARATION:The reaction of a compound of formula II (it is protected, when P contains functional groups active in the substitution reaction) with another compound of formula III (R<9> is OH, protecting group) in the presence of a base is followed by deprotection, when necessary, to give a compound of formula V. | ||||||
| 31 | Pyrazolesulfonamide derivative, production thereof and herbicide | JP29547685 | 1985-12-27 | JPS62155273A | 1987-07-10 | YAMAMOTO SUSUMU; TSUNODA TAKUYA; SATO TOSHIAKI; MORIMOTO KATSUYUKI; OYA EIICHI; IGAI TAKASHI; NAWAMAKI TSUTOMU; HATTORI KENJI |
| NEW MATERIAL:A compound expressed by formulas I {Q is formula IIWV (R 1 and R 2 are H, halogen, NO 2, alkyl, etc.; R 4 and R 7 are H, halogen or alkyl; R 6 and R 8WR 10 are H or alkyl; W 1 is O, S, etc.), etc.; m is 0W2; R is H or alkyl; B and D are R, halogen, phenyl, etc.; E is H, alkyl, etc.; W is O, S, etc.; G is formula VI [X and Y are H, alkyl, alkoxy, etc.; Z is N or CR 25 (R 25 is H, alkyl, etc.), etc.]}. EXAMPLE: N-[(4,6-Dimethoxypyrimidin-2-yl)aminocarbonyl]-1-methyl-4-(5-methyl- 1,3,4-oxadiazo-2-yl)pyrazole-5-sulfonamide. USE: A herbicide. PREPARATION: A pyrazolesulfonyl (thio)isocyanate derivative expressed by formula VII (W' is O or S) is reacted with an aminopyridine derivative expressed by formula VIII, etc., to afford the aimed compound expressed by formula I (W is W'). COPYRIGHT: (C)1987,JPO&Japio | ||||||
| 32 | 5-(3-(9-ethyl)carbazolyl)tetrazole and its production | JP18640985 | 1985-08-23 | JPS61218587A | 1986-09-29 | OKAZAKI MITSUO; YAMAGUCHI TERUHIRO; SASAKI MASAOMI |
| NEW MATERIAL:The compound of the formula. USE: A synthetic intermediate of 5-[3-(9-ethyl)carbazolyl]-1,3,4-oxadiazole derivative which is an organic photoelectric conductor. PREPARATION: The reaction of 3-cyano-9-ethylcarbazole with sodium azide is effected in an organic solvent such as methyl cellosolve to give the objective compound. COPYRIGHT: (C)1986,JPO&Japio | ||||||
| 33 | Novel 1,4-dihydropyridine derivative | JP5361485 | 1985-03-18 | JPS61212581A | 1986-09-20 | SHIMIZU NOBORU; ISHIWATARI HIROYUKI; KUNIEDA HISASHI; OTA TOMIO; ISHIHAMA HIROSHI; UCHIDA YASUYOSHI |
| NEW MATERIAL:The compound of formula I (R1 is phenyl or pyridyl which may be substituted with 1-2 halogen, nitro or CF3, or benzoxadiazolyl; R2 is lower alkyl; R3 is H, formyl, carboxyl, etc.; A is straight-chain or branched- chain lower alkylene; B is 1-6C straight-chain alkylene; X is direct bond or O). EXAMPLE:2, 6-Dimethyl-4-(3-nitrophenyl)-1, 4-dihydropyridine-3, 5-dicarboxylic acid 3-methyl ester 5-[4-(1-imidazolylmethyl)phenylmethyl] ester. USE:Vasodilator, hypotensor, antithrombotic agent and antiarteriosclerotic agent. PREPARATION:The compound of formula I can be produced by reacting the compound of formula II with N,N'-carbonyldiimidazole in an inert solvent and reacting the reaction product with the compound of formula III. | ||||||
| 34 | Acetoacetic acid ester derivative | JP2498685 | 1985-02-12 | JPS61186371A | 1986-08-20 | ONO SACHIO; MIZUKOSHI SEISHI; KOMATSU OSAMU |
| NEW MATERIAL:The acetoacetic acid ester derivative of formula I (R 1 is lower alkyl such as methyl, ethyl, propyl, isopropyl, etc., or cyclopropylmethyl). EXAMPLE: Ethyl 2-acetyl-3-(2,1,3-benzoxadiazol-4-yl)-3-bromopropionate. USE: Useful as an intermediate raw material for 1,4-dihydropyridine derivative useful pharmacologically as a vasodilator and remedy for hypertension. PREPARATION: The compound of formula I can be produced by reacting the 4-bromomethyl-benz-2,1,3-oxadiazole of formula II with the acetoacetic acid ester of formula III in the presence of a base. COPYRIGHT: (C)1986,JPO&Japio | ||||||
| 35 | JPS60501813A - | JP50287184 | 1984-07-05 | JPS60501813A | 1985-10-24 | |
| 36 | Tetrahydrobenzothiazole derivative and herbicide containing said derivative | JP6192483 | 1983-04-08 | JPS59186979A | 1984-10-23 | AOKI KATSUMICHI; SHIDA TAKAFUMI; ARAHORI HIDEO; KUMAZAWA SATOSHI; SHIMIZU SUSUMU; WATANABE TAKEO; KANDA YOUICHI; SATAKE KEIGO; YAMAZAKI SHIROU; SHINKAWA HIROE; SENDA TSUNEAKI |
| NEW MATERIAL:A tetrahydrobenzothiazole derivative of formula I (R is methyl, ethyl or propyl; R 1 is H, hydroxyl group, methoxyl group, acetoxy, propionyloxy, butyryloxy, chloroacetoxy, methoxyacetoxy, alkylamino substituted by 1W 4C alkyl group or dialkylamino; R 2 is H or together with R 1 form oxygen atoms of double bond; X is methylene, hydroxymethylene or carbonyl, etc.). EXAMPLE: 1-(5, 5-Dimethyl-4, 5, 6,7-tetrahydro-7-oxo-2-benzothiazolyl)-3-ethylimidazolidinetrione. USE: A herbicide exhibiting improved activity against gamineous and broad-leaved weeds, etc. PREPARATION: For example, a compound of formula II is reacted with glyoxal or base oxalyl, etc. to give the aimed compound of formula I . COPYRIGHT: (C)1984,JPO&Japio | ||||||
| 37 | JPS57502057A - | JP50047382 | 1981-12-14 | JPS57502057A | 1982-11-18 | |
| 38 | JPS57501480A - | JP50316181 | 1981-09-14 | JPS57501480A | 1982-08-19 | |
| 39 | 1*2*44oxadiazolinee55one derivative* its manufacture and drug composition containing same | JP14066880 | 1980-10-09 | JPS5661375A | 1981-05-26 | KAARUMAAN TAKAACHIYU; KISU AIZERUTO; ANTARU SHIMAI; PEETERU RITERAATEI NAJI; HETEIEI PATSUPU; ECHIERII PUSHIYUKAASHIYU; RAASURO SEKERESHIYU; JIYURA PATSUPU; SHIAANDORU BIRAAGU; EBUA UDOUBUARUDEI |
| 40 | JPS4985063A - | JP119873 | 1972-12-23 | JPS4985063A | 1974-08-15 | |
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