181 |
3-carbonyl having an anti-inflammatory action-1-amino-alkyl -1h- indole and its manufacturing method |
JP17305885 |
1985-08-06 |
JPH0670010B2 |
1994-09-07 |
マルコム・ライス・ベル |
|
182 |
Agricultural insecticide sterilization composition |
JP2698186 |
1986-02-12 |
JPH0662368B2 |
1994-08-17 |
昭孝 佐々木; 良雄 倉橋; 慎二 坂和; 真一 坪井; ゆみ 服部 |
PURPOSE:To obtain the titled composition exhibiting excellent insecticidal and fungicidal action and useful for the simultaneous control of blight and vermin, by using a mostly novel nitromethylene derivative with a fungicidal compound such as diisopropyl 1,3-dithiolan-2-ylidenemalnate. CONSTITUTION:The titled composition contains (A) a nitromethylene derivative of formula (X is alkyl, alkoxy or halogen; l is 0, 1 or 2; m is 2 or 3) [the compounds wherein l is 0 are known adn the others are novel: e.g. 1-(30 pyridylmethyl)-2-(nitromethylene)tetrahydropyrimidine] and (B) one or more kinds of compounds selected from diisopropyl 1,3-dithiolan-20-ylidenemalonate, 5-methyl-1,2,4-triazolo[3,4-b]benzothiazole, 3-allyloxy-1,2-benzothiazole-1,1-dioxide and 1,2,5,6-tetrahydro-4H-pyrrolo-[3,2,1-i,j]quinolin-4-one. |
183 |
Chloroacetamide derivatives |
JP1953583 |
1983-02-08 |
JPH0645617B2 |
1994-06-15 |
カ−ル・ゼツキンガ−; カ−ルハインツ・ミルツナ−; フレツド・ク−ネン |
|
184 |
Azo reroute methylamines |
JP18855883 |
1983-10-11 |
JPH0629268B2 |
1994-04-20 |
JIIKUFURIITO ETSUKURU; HANSUUGEORUKU SHUMITSUTO; BIRUFURIITO PAURUSU; HERUMAN GENTO |
|
185 |
Insecticidal nitro methylene derivative |
JP10685385 |
1985-05-21 |
JPH0629258B2 |
1994-04-20 |
SHIOKAWA KOZO; TSUBOI SHINICHI; TOSHIBE SHINZO; MORIIE KOICHI |
|
186 |
Magenta coupler - method of manufacturing |
JP18599081 |
1981-11-18 |
JPH0625135B2 |
1994-04-06 |
USAGAWA YASUSHI; NINOMYA HIDETAKA; MASUDA KOSAKU |
|
187 |
Imidazole derivative |
JP12861093 |
1993-05-31 |
JPH0649036A |
1994-02-22 |
YANAGISAWA HIROAKI; SHIMOJI YASUO; AMAMIYA YOSHIYA; KANEZAKI TAKUO; KOIKE HIROYUKI; SADA TOSHIO |
PURPOSE:To provide an imidazole derivative exhibiting excellent effect to suppress the increase of blood pressure induced by angiotensin II by oral administration and useful as a hypotensor. CONSTITUTION:The compound of formula I (R<1> is H, 1-6C alkyl; 3-6C cycloalkyl or 1-6C alkanoyl; R<2> is single bond or 1-4C alkylene; R<3> and R<4> are H or 1-6C alkyl; R<5> is H or carboxy-protecting group; R<6> is carboxy, protected carboxy or tetrazol-5-yl; X is O or S) and its pharmacologically permissible salt, e.g. 4-(1-hydroxy-1-methylethyl)-2-methoxymethyl-1-{4-[2-tetrazol-5-yl) phenyl]phenyl}methylimidazole-5-carboxylic acid methyl ester. The compound can be produced by reacting a compound of formula II with a compound of formula III in an inert solvent in the presence of a base to obtain a compound of formula IV and, as necessary, subjecting the obtained compound to reactions such as the removal of the protecting groups. |
188 |
1-Shitoroneri --5-substituted imidazo - le class |
JP5917784 |
1984-03-26 |
JPH064600B2 |
1994-01-19 |
KUWANO EIICHI; TAKEYA RITSUKO; ETO MORINOBU; ASANO MASASHI |
|
189 |
JPH0588233B2 - |
JP14455985 |
1985-07-03 |
JPH0588233B2 |
1993-12-21 |
WATANABE ISAO; MOMONOI KAISHU; HIRAIWA TOORU; ONO SATORU; NAKANO JOJI; NAGUMO KATSUYUKI; TAKAGI HIROYASU |
|
190 |
JPH0564634B2 - |
JP5361485 |
1985-03-18 |
JPH0564634B2 |
1993-09-16 |
SHIMIZU NOBORU; ISHIWATARI HIROYUKI; KUNIEDA HISASHI; OOTA TOMIO; ISHIHAMA HIROSHI; UCHIDA YASUYOSHI |
|
191 |
JPH0533716B2 - |
JP19982784 |
1984-09-25 |
JPH0533716B2 |
1993-05-20 |
TSUKAMOTO SHINICHI; TAMURA TOSHA; YOSHIDA MAKOTO; IWAMOTO HIDENORI; YAMAMOTO MINORU; KAGAMI SOICHI |
|
192 |
Intermediate compound |
JP23559091 |
1991-08-23 |
JPH0578339A |
1993-03-30 |
CRENSHAW RONNIE RAY; ALGIERI ALDO ANTONIO |
PURPOSE: To provide an intermediate for synthesis of a new 3,4- disubstituted-1,2,5-thiadiazole-1-oxide and -1,1-dioxide compd. which is an effective suppressor for the gastric acid secretion.
CONSTITUTION: The compd. of formula I [(p) is 1, 2; (n) is 2 to 4; R
2, R
3 are each H, an alkyl, alkenyl, alkynyl, cycloalkyl, amino, 2,2,2-trifluoroethyl, hydroxy, alkoxy, cyano, amidino, A'-(CH
2)
m'(CH
2)
n' (A' is phenyl, imidazoyl, thiazolyl, furyl, thienyl, etc.; m' is 0 to 2; m' is 0 to 2; n' is 2 to 4), phenyl, etc., or is, together, CH
2CH
2X(CH
2)
r ((r) is 1 to 3; X is CH
2, O, S, etc.)]. This compd. is obtd. by bringing a compd. of formula II (R
7 is eliminable, such as a halogen, phenoxy, phenylthio, alkoxy, alkylthio), and a compd. of the formula; R
10H [R
10 is NR
2R
3, NH(CH
2)
n'A'] and bringing the resulted compd. of formula III into reaction with the compd. of formula HS(CH
2)
nNH
2.
COPYRIGHT: (C)1993,JPO |
193 |
JPH0510345B2 - |
JP1856484 |
1984-02-03 |
JPH0510345B2 |
1993-02-09 |
MAKIKADO TOKUO; MURABAYASHI AKIRA; HATSUTA TAKAYUKI; ISHIGURO TAKEO |
|
194 |
JPH0460114B2 - |
JP7296684 |
1984-04-13 |
JPH0460114B2 |
1992-09-25 |
SHIOKAWA KOZO; TSUBOI SHINICHI; TOSHIBE SHINZO; MORIIE KOICHI |
|
195 |
JPH0432061B2 - |
JP13108583 |
1983-07-20 |
JPH0432061B2 |
1992-05-28 |
|
|
196 |
JPH0415781B2 - |
JP16395183 |
1983-09-05 |
JPH0415781B2 |
1992-03-19 |
TSURUTA MINEO; OOE TAKANORI; KAWASAKI KAZUYUKI; MIKASHIMA HIROSHI; YASUDA HIROSHI |
|
197 |
JPH0374663B2 - |
JP19732984 |
1984-09-20 |
JPH0374663B2 |
1991-11-27 |
|
|
198 |
JPH0374227B2 - |
JP4834784 |
1984-03-14 |
JPH0374227B2 |
1991-11-26 |
|
|
199 |
JPH0329077B2 - |
JP16725984 |
1984-08-09 |
JPH0329077B2 |
1991-04-23 |
URUSU BURUTSUKUHARUTO |
|
200 |
JPH0324448B2 - |
JP23387885 |
1985-10-19 |
JPH0324448B2 |
1991-04-03 |
SEO AKIRA; SUGANO HIDEO; HASEGAWA NOBORU; IKEDA KENICHI; MUNECHIKA YUKIMI; OMI TETSUTO; KONAKA SHIGEO; UCHIDA MATAZAEMON |
|