首页 / 专利分类库 / 有机化学 / 杂环化合物 / 杂环化合物,含1,3-二唑或氢化1,3-二唑环、不与其他环稠合
序号 专利名 申请号 申请日 公开(公告)号 公开(公告)日 发明人
181 3-carbonyl having an anti-inflammatory action-1-amino-alkyl -1h- indole and its manufacturing method JP17305885 1985-08-06 JPH0670010B2 1994-09-07 マルコム・ライス・ベル
182 Agricultural insecticide sterilization composition JP2698186 1986-02-12 JPH0662368B2 1994-08-17 昭孝 佐々木; 良雄 倉橋; 慎二 坂和; 真一 坪井; ゆみ 服部
PURPOSE:To obtain the titled composition exhibiting excellent insecticidal and fungicidal action and useful for the simultaneous control of blight and vermin, by using a mostly novel nitromethylene derivative with a fungicidal compound such as diisopropyl 1,3-dithiolan-2-ylidenemalnate. CONSTITUTION:The titled composition contains (A) a nitromethylene derivative of formula (X is alkyl, alkoxy or halogen; l is 0, 1 or 2; m is 2 or 3) [the compounds wherein l is 0 are known adn the others are novel: e.g. 1-(30 pyridylmethyl)-2-(nitromethylene)tetrahydropyrimidine] and (B) one or more kinds of compounds selected from diisopropyl 1,3-dithiolan-20-ylidenemalonate, 5-methyl-1,2,4-triazolo[3,4-b]benzothiazole, 3-allyloxy-1,2-benzothiazole-1,1-dioxide and 1,2,5,6-tetrahydro-4H-pyrrolo-[3,2,1-i,j]quinolin-4-one.
183 Chloroacetamide derivatives JP1953583 1983-02-08 JPH0645617B2 1994-06-15 カ−ル・ゼツキンガ−; カ−ルハインツ・ミルツナ−; フレツド・ク−ネン
184 Azo reroute methylamines JP18855883 1983-10-11 JPH0629268B2 1994-04-20 JIIKUFURIITO ETSUKURU; HANSUUGEORUKU SHUMITSUTO; BIRUFURIITO PAURUSU; HERUMAN GENTO
185 Insecticidal nitro methylene derivative JP10685385 1985-05-21 JPH0629258B2 1994-04-20 SHIOKAWA KOZO; TSUBOI SHINICHI; TOSHIBE SHINZO; MORIIE KOICHI
186 Magenta coupler - method of manufacturing JP18599081 1981-11-18 JPH0625135B2 1994-04-06 USAGAWA YASUSHI; NINOMYA HIDETAKA; MASUDA KOSAKU
187 Imidazole derivative JP12861093 1993-05-31 JPH0649036A 1994-02-22 YANAGISAWA HIROAKI; SHIMOJI YASUO; AMAMIYA YOSHIYA; KANEZAKI TAKUO; KOIKE HIROYUKI; SADA TOSHIO
PURPOSE:To provide an imidazole derivative exhibiting excellent effect to suppress the increase of blood pressure induced by angiotensin II by oral administration and useful as a hypotensor. CONSTITUTION:The compound of formula I (R<1> is H, 1-6C alkyl; 3-6C cycloalkyl or 1-6C alkanoyl; R<2> is single bond or 1-4C alkylene; R<3> and R<4> are H or 1-6C alkyl; R<5> is H or carboxy-protecting group; R<6> is carboxy, protected carboxy or tetrazol-5-yl; X is O or S) and its pharmacologically permissible salt, e.g. 4-(1-hydroxy-1-methylethyl)-2-methoxymethyl-1-{4-[2-tetrazol-5-yl) phenyl]phenyl}methylimidazole-5-carboxylic acid methyl ester. The compound can be produced by reacting a compound of formula II with a compound of formula III in an inert solvent in the presence of a base to obtain a compound of formula IV and, as necessary, subjecting the obtained compound to reactions such as the removal of the protecting groups.
188 1-Shitoroneri --5-substituted imidazo - le class JP5917784 1984-03-26 JPH064600B2 1994-01-19 KUWANO EIICHI; TAKEYA RITSUKO; ETO MORINOBU; ASANO MASASHI
189 JPH0588233B2 - JP14455985 1985-07-03 JPH0588233B2 1993-12-21 WATANABE ISAO; MOMONOI KAISHU; HIRAIWA TOORU; ONO SATORU; NAKANO JOJI; NAGUMO KATSUYUKI; TAKAGI HIROYASU
190 JPH0564634B2 - JP5361485 1985-03-18 JPH0564634B2 1993-09-16 SHIMIZU NOBORU; ISHIWATARI HIROYUKI; KUNIEDA HISASHI; OOTA TOMIO; ISHIHAMA HIROSHI; UCHIDA YASUYOSHI
191 JPH0533716B2 - JP19982784 1984-09-25 JPH0533716B2 1993-05-20 TSUKAMOTO SHINICHI; TAMURA TOSHA; YOSHIDA MAKOTO; IWAMOTO HIDENORI; YAMAMOTO MINORU; KAGAMI SOICHI
192 Intermediate compound JP23559091 1991-08-23 JPH0578339A 1993-03-30 CRENSHAW RONNIE RAY; ALGIERI ALDO ANTONIO
PURPOSE: To provide an intermediate for synthesis of a new 3,4- disubstituted-1,2,5-thiadiazole-1-oxide and -1,1-dioxide compd. which is an effective suppressor for the gastric acid secretion. CONSTITUTION: The compd. of formula I [(p) is 1, 2; (n) is 2 to 4; R 2, R 3 are each H, an alkyl, alkenyl, alkynyl, cycloalkyl, amino, 2,2,2-trifluoroethyl, hydroxy, alkoxy, cyano, amidino, A'-(CH 2) m'(CH 2) n' (A' is phenyl, imidazoyl, thiazolyl, furyl, thienyl, etc.; m' is 0 to 2; m' is 0 to 2; n' is 2 to 4), phenyl, etc., or is, together, CH 2CH 2X(CH 2) r ((r) is 1 to 3; X is CH 2, O, S, etc.)]. This compd. is obtd. by bringing a compd. of formula II (R 7 is eliminable, such as a halogen, phenoxy, phenylthio, alkoxy, alkylthio), and a compd. of the formula; R 10H [R 10 is NR 2R 3, NH(CH 2) n'A'] and bringing the resulted compd. of formula III into reaction with the compd. of formula HS(CH 2) nNH 2. COPYRIGHT: (C)1993,JPO
193 JPH0510345B2 - JP1856484 1984-02-03 JPH0510345B2 1993-02-09 MAKIKADO TOKUO; MURABAYASHI AKIRA; HATSUTA TAKAYUKI; ISHIGURO TAKEO
194 JPH0460114B2 - JP7296684 1984-04-13 JPH0460114B2 1992-09-25 SHIOKAWA KOZO; TSUBOI SHINICHI; TOSHIBE SHINZO; MORIIE KOICHI
195 JPH0432061B2 - JP13108583 1983-07-20 JPH0432061B2 1992-05-28
196 JPH0415781B2 - JP16395183 1983-09-05 JPH0415781B2 1992-03-19 TSURUTA MINEO; OOE TAKANORI; KAWASAKI KAZUYUKI; MIKASHIMA HIROSHI; YASUDA HIROSHI
197 JPH0374663B2 - JP19732984 1984-09-20 JPH0374663B2 1991-11-27
198 JPH0374227B2 - JP4834784 1984-03-14 JPH0374227B2 1991-11-26
199 JPH0329077B2 - JP16725984 1984-08-09 JPH0329077B2 1991-04-23 URUSU BURUTSUKUHARUTO
200 JPH0324448B2 - JP23387885 1985-10-19 JPH0324448B2 1991-04-03 SEO AKIRA; SUGANO HIDEO; HASEGAWA NOBORU; IKEDA KENICHI; MUNECHIKA YUKIMI; OMI TETSUTO; KONAKA SHIGEO; UCHIDA MATAZAEMON
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